2024年5月7日发(作者：冷书文)
2(CH2)2C＝
NOiPr H Cl 1.171> C2H5 H H
0(CH2)2C＝
NOCH2CH＝
CHCl
H Cl
1.172> C2H5 H H
2(CH2)2C＝
NOCH2CH＝
CHCl
H Cl
1.173> C2H5 H H
0(CH2)2C＝
NOCH2C6H5
H
Cl 1.174 C2H5>
H H 2(CH2ub>)2
C＝
NOCH2C6H5 H
Cl 1.175 C2H5>
H H 0(CH2ub>)2
C(CH3)2
H Cl 1.176 C2b>H5
H H 2y>(CH2)2C(CH3)2
H Cl
1.177ry> CH3 CH3 Hry> 0(CH2)2C＝
O H CH3
>lspec> 序号 R15 R16 R<sup>17
n X Y L M
1.178> CH3 CH3 H> 2(CH2)2C＝
O H CH3
1.179
CH3 CH3> H 0(CH2)2
CHOCH3 H CH3
ow> 1.180 CH3 CH3
H 2(CH2)2<
/sub>CHOCH3 H CHb>3
1.181 CH3y> CH3 H 0(CH<
sub>2)2
CHOC2H5y> H CH3
1.182ntry> CH3 CH3 Hntry> 2(CH2)2CHOC
2H5
H CH3try>
1.183 CH3 CH3
H 0(CH2)<sub>2
CHOiPr H CH3b>
1.184 CH3y> CH3 H 2(CH2sub>)2
CHOiPr H CH>3
1.185 CH3> CH3 H 0(CHub>2)2
CHOH H C
H3
1.186 CH3 CH3 H 2(CH2)2
CHOH Htry> CH3
1.187 CH3 CH3 H 0<entry>(CH2)2C＝
NOCH3 H CH3
w> 1.188 CH3 CH3<
/sub> H 2(CH2)2ub>
C＝
NOCH3 H CH3
w> 1.189 CH3 CH3<
/sub> H 0(CH2)2ub>
C＝
NOC2H5 H CH3>
1.190 CH3> CH3 H 2(CH2ub>)2
C＝
NOC2H5 H CH3>
1.191 CH3> CH3 H 0(CH2ub>)2
C＝
NOiPr H CH3
y> 1.192 CH3 CH3
H 2(CH2)2<
entry>C＝
NOiPr H CH3
|
y> 1.193 CH3 CH3
H 0(CH2)2<
entry>C＝NOCH2CH＝
CHCl H CH3
|
> 1.194 CH3 CH3ntry> H 2(CH2)2try>C＝NOCH2CH＝
CHCl H CH3
|
> 1.195 CH3 CH3ntry> H 0(CH2)2try>C＝
NOCH2C6H5 H
CH3
|
1.196 CH3b>
CH3 H 2y>(CH2)2C＝
NOCH2C6H5 H
CH3
1.197 CH3b>
CH3 H 0y>(CH2)2C(CH3)2
H CH3
1.198
CH3 CH3 H
2(CH2)2C(CH3)2
H CH3</entry>
1.199 C2H5ntry> H H 0(CH2)
2
C＝O
H CH3
1.200
C2H5 H H
2(CH2)2C＝
O
H CH3
1.201
C2H5 H H
0(CH2)2CHOCH3
H CH3w> 1.202 C2H5> H H 2(CH2)2b>
CHOCH3 H CH3
1.203 C2H5sub>
H H 0(CH2
)2CHOC2H5ry> H CH3
1.204ntry> C2H5 H Hry> 2(CH2)2CHOC2sub>H5
H CH3
w> 1.205 C2H5> H H 0(CH2)2b>
CHOiPr H CH3
>
1.206 C2H5
H H 2(CH2)>2
CHOiPr H CH3
1.207 C2H5entry> H H 0(CH2
)2
CHOH H CH3ub>
1.208 C2H5>
H H 2(CH2ub>)2
CHOH H CH3
1.209 C2H5 H H 0(CH>2)2
C＝NOCH3
H CH3w> 1.210 C2H5> H H 2(CH2)2b>
C＝
NOCH3 H CH3
w> 1.211 C2H5> H H 0(CH2)2b>
C＝
NOC2H5 H CH3>
1.212 C2H5
H H 2(CH2b>)2
C＝
NOC2H5 H CH3>
1.213 C2H5
H H 0(CH2b>)2
C＝
NOiPr H CH3
y> 1.214 C2H5 Hntry> H 2(CH2)2try>C＝
NOiPr H CH3
|
group>
c> 序号 R15 R16 R<sup>17
n X Y L M
1.215> C2H5 H H
0(CH2)2C＝
NOCH2CH＝
CHCl H CH3
> 1.216 C2H5 Htry> H2(CH2)2y>C＝NOCH2CH＝
CHCl H CH3
|
> 1.217 C2H5 Htry> H0(CH2)2y>C＝
NOCH2C6H5 H
CH3
|
1.218 C2H5
H H2(CH2)2
C＝NOCH2C6H5
H CH3
1.219 C2H5
H H0(CH2)2
C(CH3)2ntry> H CH3
1.220 C2H5 H Hentry>2(CH2)2C(CH
3)2
H CH3ry>
1.221 CH3 CH<sub>3
p-CH3-C6H4-SO2-
0(CH2)2C＝O
H CH3
1.222
CH3 CH3> p-CH3-C6H4-SO2-
2(CH2)2C＝
O H CH3
1.223
CH3 CH3> p-CH3-C6H4-SO2-
0(CH2)2CH
OCH3 H CH3
> 1.224 CH3 CH3ub>
p-CH3-C6H4-
SO2-
2(CH2)2CH
OCH3 H CH3
> 1.225 CH3 CH3ub>
p-CH3-C6H4-
SO2-
0(CH2)2CH
OC2H5 H CH3
1.226 CH3 CH3
p-CH3-C6H4-SO2-
2(CH2)2CHOC2H5
H CH3
1.227 CH3 CH3
P-CH3-C6H4-SO2-
0(CH2)2CHOiPr
H CH3
1.228
CH3 CH3try> p-CH3-C6H4-SO2-
2(CH2)2CH
OiPr H CH3
|
1.229
CH3 CH3try> p-CH3-C6H4-SO2-
0(CH2)2CH
OH H CH3
|
1.230
CH3 CH3ry> P-CH3-C6H4-SC2-
2(CH2)2CH
OH H CH3
1.231
CH3 CH3ry> p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH3 H CH3
w> 1.232 CH3 CH3<
/sub> p-CH3-C6H4-
SO2-
2(CH2)2C＝
NOCH3 H CH3
w> 1.233 CH3 CH3<
/sub> p-CH3-C6H4-
SO2-
0(CH2)2C＝
NOC2H5 H CH3>
1.234 CH3> CH3 p-CH3-
C6H4-SO2-
2(CH2)2C＝
NOC2H5 H CH3>
1.235 CH3> CH3 p-CH3-
C6H4-SO2-
0(CH2)2C＝
NOiPr H CH3
y> 1.236 CH3 CH3
p-CH3-C6H4-SO2-
2(CH2)2C＝
NOiPr H CH3
|
y> 1.237 CH3 CH3
p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH2CH＝
CHCl H CH3
|
> 1.238 CH3 CH3ntry> p-CH3-C6H4-SO2-
2(CH2)2C＝
NOCH2CH＝
CHCl H CH3
|
> 1.239 CH3 CH3ntry> p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH2C6H5 H
CH3
|
1.240 CH3b>
CH3 p-CH3-C6H4-SO2-
2(CH2)2C＝NOCH2C6H5
H CH3
1.241 CH3b>
CH3 p-CH3-C6H4-SO2-
0(CH2)2C(CH3)2
H CH3ntry>
1.242 CH3 CH3
p-CH3-C6H4-SO2-
2(CH2)2C(CH3)2
H CH3ntry>
1.243 C2H5ry> H p-CH3-C6H4-
SO2-
0(CH2)2C＝O
H CH3
1.244
C2H5 H p-CH3-C6H4-SO2-
2(CH2)2C＝O
H CH3
1.245
C2H5 H p-CH3-C6H4-SO2-
0(CH2)2CHOCH3
H CH3> 1.246 C2H5
H p-CH3-C6H4-
SO2-
2(CH2)2CH
OCH3 H CH3
> 1.247 C2H5
H p-CH3-C6H4-
SC2-
0(CH2)2CH
OC2H5 H CH3
1.248 C2H5entry> H p-CH3-C6H4-
SO2-
2(CH2)2CHOC2H5
H CH3
1.249 C2H5entry> H p-CH3-C6H4-
SO2-
0(CH2)2CHOiPr
H CH3
1.250
C2H5 Hy> p-CH3-C6H4-SO2-
2(CH2)2CH
OiPr H CH3
|
1.251
C2H5 Hy> p-CH3-C6H4-SO2-
0(CH2)2CH
OH H CH3
|
up>
<colspec> 序号R15 R16 R<sup>17
n X Y L M
1.252> C2H5 H p-
CH3-C6H4-SO2-
2(CH2)2CH
OH H CH3
1.253
C2H5 H> p-CH3-C6H4-SO2-
0(CH2)2C
＝
NOCH3 H CH3
w> 1.254 C2H5> H p-CH3-C6H4-
SO2-
2(CH2)2C
＝
NOCH3 H CH3
w> 1.255 C2H5> H p-CH3-C6H4-
SO2-
0(CH2)2C
＝
NOC2H5 H CH3>
1.256 C2H5
H p-CH3-
C6H4-SO2-
2(CH2)2C
＝
NOC2H5 H CH3>
1.257 C2H5
H p-CH3-
C6H4-SO2-
0(CH2)2C
＝
NOiPr H CH3
y> 1.258 C2H5 Hntry> p-CH3-C6H4-SO2-
2(CH2)2C
＝
NOiPr H CH3
|
y> 1.259 C2H5 Hntry> p-CH3-C6H4-SO2-
0(CH2)2C
＝NOCH2CH＝
CHCl H CH3
|
> 1.260 C2H5 Htry> p-CH3-C6H4-SO2-
2(CH2)2C
＝NOCH2CH＝
CHCl H CH3
|
> 1.261 C2H5 Htry> p-CH3-C6H4-SO2-
0(CH2)2C
＝
NOCH2C6H5 H
CH3
|
1.262 C2H5
H p-CH3-C6H4-SO2-
2(CH2)2C＝
NOCH2C6H5
H CH3
1.263 C2H5
H p-CH3-C6H4-SO2-
0(CH2)2C(CH3)2
H CH3entry>
1.264 C2H5try> H P-CH3-C6H4-
SO2-
2(CH2)2C(CH3)2
H CH3entry>
1.265 CH3 CH3
H 0 CH2CH-NHCH3
H H
> 1.266 CH3 CH3ntry> H 2 CH2CH-
NHCH3 H H
|
> 1.267 CH3 CH3ntry> H 0 CH2CH-
NHC2H5 H H
> 1.268 CH3 CH3ub>
H 2 CH2ry>CH-
NHC2H5 H H
> 1.269 CH3 CH3ub>
H 0 CH2ry>CH-
N(CH3)2 H H
> 1.270 CH3 CH3ub>
H 2 CH2ry>CH-
N(CH3)2 H H
> 1.271 CH3 CH3ub>
H 0 CH2ry>CH-
NHOC2H5 H H
w> 1.272 CH3 CH3<
/sub> H 2 CH2ntry>CH-
NHOC2H5 H H
w> 1.273 CH3 CH3<
/sub> H 0 CH2ntry>CH-
N(CH3)OC2H5 Hy> H
1.274 CH3ntry> CH3 H 2 CH2
CH-
N(CH3)OC2H5 Hy> H
1.275 CH3ntry> CH3 H 0 CH2
C＝N-
NH2 H H
1
.276 CH3 CH3y> H 2 CH2C＝N-
NH2 H H
1
.277 CH3 CH3y> H 0 CH2C＝N-
N(CH3)2 H H
> 1.278 CH3 CH3ub>
H 2 CH2ry>C＝N-
N(CH3)2 H H
> 1.279 CH3 CH3ub>
H 0 CH2ry>C(CH3)-
OCH3 H H
1.280 CH3 CH3ry> H 2 CH2C(CH3
)-
OCH3 H H
1.281 CH3 CH3ry> H 0 CH2Ontry> H H
1.282 CHb>3
CH3 H 2y> CH2O H H
ntry>
|
1.283 C2H5ry> H H 0 CH2ntry>CH-
NHCH3
H H
> 1.284 C2H5 Htry> H 2 CH2CH-
NHCH3 H H
|
> 1.285 C2H5 Htry> H 0 CH2CH-
NHC2H5 H H
> 1.286 C2H5
H H 2 CH2>CH-
NHC2H5 H H
> 1.287 C2H5
H H 0 CH2>CH-
N(CH3)2 H H
> 1.288 C2H5
H H 2 CH2>CH-
N(CH3)2 H H
>
|
spec>> 序号
R15 R16 R<
sup>17 n X Y L
M
|
1.289> C2H5 H H
0 CH2 CH-
NHOC2H5 H H
w> 1.290 C2H5> H H 2 CH2ry> CH-
NHOC2H5 H H
w> 1.291 C2H5> H H 0 CH2ry> CH-
N(CH3)OC2H5 Hy> H
1.292 C2H5b>
H H 2 CH2sub>
CH-
N(CH3)OC2H5 Hy> H
1.293 C2H5b>
H H 0 CH2sub>
C＝N-
NH2 H H
1.294
C2H5 H H
2 CH2 C＝N-NH2
H H
1.295
C2H5 H H
0 CH2 C＝N-N(CH3)2
H H> 1.296 C2H5
H H 2 CH2> C＝N-
N(CH3)2 H H
> 1.297 C2H5
H H 0 CH2> C(CH3)-
OCH3 H H
1.298
C2H5 H> H 2 CH2 C(CH3<
/sub>)-
OCH3 H H
1.299
C2H5 H> H 0 CH2 Ory> H H
1.300 C2H5 H H 2<entry> CH2 O H H>
1.301 CH3 CHb>3
H 0 CH2y> CH-
NHCH3
H CH3w> 1.302 CH3 CH3<
/sub> H 2 CH2ntry> CH-
NHCH3 H CH3
w> 1.303 CH3 CH3<
/sub> H 0 CH2ntry> CH-
NHC2H5 H CH3>
1.304 CH3> CH3 H 2 CH2ub>
CH-
NHC2H5 H CH3>
1.305 CH3> CH3 H 0 CH2ub>
CH-
N(CH3)2 H CH3>
1.306 CH3> CH3 H 2 CH2ub>
CH-
N(CH3)2 H CH3>
1.307 CH3> CH3 H 0 CH2ub>
CH-
NHOC2H5 H CH3b>
1.308 CH3y> CH3 H 2 CH2sub>
CH-
NHOC2H5 H CH3b>
1.309 CH3y> CH3 H 0 CH2sub>
CH-
N(CH3)OC2H5 Hy> CH3
1.310 CH3sub>
CH3 H 2ntry> CH2 CH-
N(CH3)OC2H5 Hy> CH3
1.311 CH3sub>
CH3 H 0ntry> CH2 C＝N-
NH2 H CH3
<row> 1.312 CH3 CH3>
H 2 CH2> C＝N-
NH2 H CH3<
row> 1.313 CH3 CH3>
H 0 CH2> C＝N-
N(CH3)2 H CH3>
1.314 CH3> CH3 H 2 CH2ub>
C＝N-
N(CH3)2 H CH3>
1.315 CH3> CH3 H 0 CH2ub>
C(CH3)-
OCH3 H CH3
> 1.316 CH3 CH3ub>
H 2 CH2ry> C(CH3)-
OCH3 H CH3
> 1.317 CH3 CH3ub>
H 0 CH2ry> O H CH3
> 1.318 CH3 CH3ntry> H 2 CH2 O
H CH3
|
1.319y> C2H5 H H
> 0 CH2 CH-
NHCH3 H CH3
w> 1.320 C2H5> H H 2 CH2ry> CH-
NHCH3 H CH3
w> 1.321 C2H5> H H 0 CH2ry> CH-
NHC2H5 H CH3>
1.322 C2H5
H H 2 CH2b>
CH-
NHC2H5 H CH3>
1.323 C2H5
H H 0 CH2b>
CH-
N(CH3)2 H CH3>
1.324 C2H5
H H 2 CH2b>
CH-
N(CH3)2 H CH3>
1.325 C2H5
H H 0 CH2b>
CH-
NHOC2H5 H CH3b>
c>ad> 序号
R15 R16 R<
sup>17 n X Y L
M
1.326> C2H5 H H
2 CH2 CH-
NHOC2H5 H CH3b>
1.327 C2H5>
H H 0 CH2ub>
CH-N(CH3)OC2H5
Hy> CH3
1.328 C2b>H5
H H 2y> CH2 CH-
N(CH3)OC2H5 Hy> CH3
1.329 C2b>H5
H H 0y> CH2 C＝N-
NH2 H CH3
<row> 1.330 C2H5 H
H2 CH2
C＝N-
NH2 H CH3<
row> 1.331 C2H5 H
H 0 CH2
C＝N-
N(CH3)2 H CH3>
1.332 C2H5
H H 2 CH2b>
C＝N-
N(CH3)2 H CH3>
1.333 C2H5
H H 0 CH2b>
C(CH3)-
OCH3 H CH3
> 1.334 C2H5
H H 2 CH2> C(CH3)-
OCH3 H CH3
> 1.335 C2H5
H H 0 CH2> O H CH3
1.336 C2H5 Hy> H 2 CH2 Ontry> H CH3 1.337
CH3 CH3 H
0 CH2 CH-
NHCH3 H Cl> 1.338 CH3 CH3ntry> H 2 CH2 CH-
NHCH3 H Cl
|
> 1.339 CH3 CH3ntry> H 0 CH2 CH-
NHC2H5 H Cl
> 1.340 CH3 CH3ub>
H 2 CH2ry> CH-
NHC2H5 H Cl
> 1.341 CH3 CH3ub>
H 0 CH2ry> CH-
N(CH3)2 H Cl
> 1.342 CH3 CH3ub>
H 2 CH2ry> CH-
N(CH3)2 H Cl
> 1.343 CH3 CH3ub>
H 0 CH2ry> CH-
NHOC2H5 H Cl
w> 1.344 CH3 CH3<
/sub> H 2 CH2ntry> CH-
NHOC2H5 H Cl
w> 1.345 CH3 CH3<
/sub> H 0 CH2ntry> CH-
N(CH3)OC2H5 Hy> Cl
1.346 CH3ntry> CH3 H 2 CH2
CH-
N(CH3)OC2H5 Hy> Cl
1.347 CH3ntry> CH3 H 0 CH2
C＝N-
NH2 H Cl
1
.348 CH3 CH3y> H 2 CH2 C＝N-
NH2 H Cl
1
.349 CH3 CH3y> H 0 CH2 C＝N-
N(CH3)2 H Cl
> 1.350 CH3 CH3ub>
H 2 CH2ry> C＝N-
N(CH3)2 H Cl
> 1.351 CH3 CH3ub>
H 0 CH2ry> C(CH3)-
OCH3 H Cl
1.352 CH3 CH3ry> H 2 CH2 C(CH
3)-
OCH3 H Cl
1.353 CH3 CH3ry> H 0 CH2 Ontry> H Cl
1.354 CHb>3
CH3 H 2
|
y> CH2 O H Clentry> 1.355 C2H5try> H H 0 CH2entry> CH-
NHCH3
H Cl
> 1.356
|
C2H5 Htry> H 2 CH2 CH-
NHCH3 H Cl> 1.357 C2H5 Htry> H 0 CH2 CH-
NHC2H5 H Cl
> 1.358 C2H5
H H 2 CH2> CH-
NHC2H5 H Cl
> 1.359 C2H5
H H 0 CH2> CH-
N(CH3)2 H Cl
> 1.360 C2H5
H H 2 CH2> CH-
N(CH3)2 H Cl
> 1.361 C2H5
H H 0 CH2> CH-
NHOC2H5 H Cl
w> 1.362 C2H5> H H 2 CH2ry> CH-
NHOC2H5 H Cl
w>
|
olspec>y> 序号
R15 R16 R<
sup>17 n X Y L
M
|
1.363> C2H5 H H
0 CH2 CH-
N(CH3)OC2H5 Hy> Cl
1.364 C2H5ub>
H H 2 CH2 CH-N(CH3)OC2H5
Hy> Cl
1.365 C2H5ub>
H H 0 CH2 C＝N-NH2
H Cl
1.366
C2H5 H H
2 CH2 C＝N-NH2
H Cl
1.367
C2H5 H H
0 CH2 C＝N-N(CH3)2
H Cl> 1.368 C2H5
H H 2 CH2> C＝N-
N(CH3)2 H Cl
> 1.369 C2H5
H H 0 CH2> C(CH3)-
OCH3 H Cl
1.370
C2H5 Hy> H 2 CH2 C(CH3
)-
OCH3 H Cl
1.371
C2H5 Hy> H 0 CH2 Ontry> H Cl
1.372 C>2H5
H H 2> CH2 O H Clntry>
1.373 CH3 CH3
H 0(CH2)2
CH-NHCH3
H H
> 1.374 CH3 CH3ntry> H 2(CH2)2try> CH-
NHCH3 H H
|
> 1.375 CH3 CH3ntry> H 0(CH2)2try> CH-
NHC2H5 H H
> 1.376 CH3 CH3ub>
H 2(CH2)2b>
CH-
NHC2H5 H H
> 1.377 CH3 CH3ub>
H 0(CH2)2b>
CH-
N(CH3)2 H H
> 1.378 CH3 CH3ub>
H 2(CH2)2b>
CH-
N(CH3)2 H H
> 1.379 CH3 CH3ub>
H 0(CH2)2b>
CH-
NHOC2H5 H H
w> 1.380 CH3 CH3<
/sub> H 2(CH2)2ub>
CH-
NHOC2H5 H H
w> 1.381 CH3 CH3<
/sub> H 0(CH2)2ub>
CH-
N(CH3)OC2H5 Hy> H
|
1.382 CH3ntry> CH3 H 2(CH
2)2 CH-
N(CH3)OC2H5 Hy> H
1.383 CH3ntry> CH3 H 0(CH
2)2 C＝N-
NH2 H H
1.384
CH3 CH3y> H 2(CH2)2> C＝N-
NH2 H H
1.385
CH3 CH3y> H 0(CH2)2> C＝N-
N(CH3)2 H H
> 1.386 CH3 CH3ub>
H 2(CH2)2b>
C＝N-
N(CH3)2 H H
> 1.387 CH3 CH3ub>
H 0(CH2)2b>
C(CH3)-
OCH3 H H
1.388
CH3 CH3ry> H 2(CH2)2y> C(CH3)-
OCH3 H H
1.389
CH3 CH3ry> H 0(CH2)2y> O H H
1.390 CH3 CH3 H
2(CH2)2 O<
entry> H H
1.391 C>2H5
H H 0>(CH2)2 CH-
NHCH3
H H
> 1.392 C2H5 Htry> H 2(CH2)2y> CH-
NHCH3 H H
|
> 1.393 C2H5 Htry> H 0(CH2)2y> CH-
NHC2H5 H H
> 1.394 C2H5
H H 2(CH2)2>
CH-
NHC2H5 H H
> 1.395 C2H5
H H 0(CH2)2>
CH-
N(CH3)2 H H
> 1.396 C2H5
H H 2(CH2)2>
CH-
N(CH3)2 H H
> 1.397 C2H5
H H 0(CH2)2>
CH-
NHOC2H5 H H
w> 1.398 C2H5> H H 2(CH2)2b>
CH-
NHOC2H5 H H
w> 1.399 C2H5> H H 0(CH2)2b>
CH-
N(CH3)OC2H5 Hy> H
|
pec>head> 序号
R15 R16 R<
sup>17 n XY L
M
1.400> C2H5 H H
2(CH2)2CH-
N(CH3)OC2H5 Hy> H
1.401 C2H5b>
H H 0(CH2sub>)2
C＝N-NH2
H H
1.402
C2H5 H H
2(CH2)2C＝N-
NH2
H H
1.403
C2H5 H H
0(CH2)2C＝N-
N(CH3)2
H H> 1.404 C2H5
H H 2(CH2)2>
C＝N-
N(CH3)2 H H
> 1.405 C2H5
H H 0(CH2)2>
C(CH3)-
OCH3 H H
1.406
C2H5 H> H 2(CH2)2
C(CH3)-
OCH3 H H
1.407
C2H5 H> H 0(CH2)2
O H H
1.408try> C2H5 H Hy> 2(CH2)2O> H H
1.409 CH3 CH3 H 0<entry>(CH2)2CH-
NHCH3 H CH3
w> 1.410 CH3 CH3> H 2(CH2)2
CH-
NHCH3
H CH3w> 1.411 CH3 CH3<
/sub> H 0(CH2)2ub>
CH-
NHC2H5 H CH3>
1.412 CH3> CH3 H 2(CH2ub>)2
CH-
NHC2H5 H CH3>
1.413 CH3> CH3 H 0(CH2ub>)2
CH-
N(CH3)2 H CH3>
1.414 CH3> CH3 H 2(CH2ub>)2
CH-
N(CH3)2 H CH3>
1.415 CH3> CH3 H 0(CH2ub>)2
CH-
NHOC2H5 H CH3b>
1.416 CH3y> CH3 H 2(CH2sub>)2
CH-
NHOC2H5 H CH3b>
1.417 CH3y> CH3 H 0(CH2sub>)2
CH-
N(CH3)OC2H5 Hy> CH3
1.418 CH3sub>
CH3 H 2ntry>(CH2)2CH-
N(CH3)OC2H5 Hy> CH3
1.419 CH3sub>
CH3 H 0ntry>(CH2)2C＝N-
NH2 H CH3
<
row> 1.420 CH3 CH3>
H 2(CH2)2
C＝N-
NH2 H CH3
<row> 1.421 CH3 CH3>
H 0(CH2)2
C＝N-
N(CH3)2 H CH3>
1.422 CH3> CH3 H 2(CH2ub>)2
C＝N-
N(CH3)2 H CH3>
1.423 CH3> CH3 H 0(CH2ub>)2
C(CH3)-
OCH3 H CH3
> 1.424 CH3 CH3ub>
H 2(CH2)2b>
C(CH3)-
OCH3 H CH3
> 1.425 CH3 CH3ub>
H 0(CH2)2b>
O H CH3> 1.426 CH3 CH3ub>
H 2(CH2)2b>
O H CH3> 1.427 C2H5
H H 0(CH2)2>
CH-
NHCH3 H CH3
w> 1.428 C2H5> H H 2(CH2)2b>
CH-
NHCH3 H CH3
w> 1.429 C2H5> H H 0(CH2)2b>
CH-
NHC2H5 H CH3>
1.430 C2H5
H H 2(CH2b>)2
CH-
NHC2H5 H CH3>
1.431 C2H5
H H 0(CH2b>)2
CH-
N(CH3)2 H CH3>
1.432 C2H5
H H 2(CH2b>)2
CH-
N(CH3)2 H CH3>
1.433 C2H5
H H 0(CH2b>)2
CH-
NHOC2H5 H CH3b>
1.434 C2H5>
H H 2(CH2ub>)2
CH-
NHOC2H5 H CH3b>
1.435 C2H5>
H H 0(CH2ub>)2
CH-
N(CH3)OC2H5 Hy> CH3 1.436 C2b>H5
H H 2y>(CH2)2CH-
N(CH3)OC2H5 Hy> CH3
>ec> 序号 R15 R16 R<sup>17
n XY L M
1.437> C2H5 H H
0(CH2)2C＝N-
NH2 H CH3
<row> 1.438 C2H5 H
H 2(CH2)2<
/entry>C＝N-
NH2 H CH3<
row> 1.439 C2H5 H
H 0(CH2)2<
/entry>C＝N-
N(CH3)2 H CH3>
1.440 C2H5
H H 2(CH2b>)2
C＝N-
N(CH3)2 H CH3>
1.441 C2H5
H H 0(CH2b>)2
C(CH3)-
OCH3 H CH3
> 1.442 C2H5
H H 2(CH2)2>
C(CH3)-
OCH3 H CH3
> 1.443 C2H5
H H 0(CH2)2>
O H CH3
> 1.444 C2H5
H H 2(CH2)2>
O H CH3
> 1.445 CH3 CH3ub>
H 0(CH2)2b>
CH-
NHCH3 H Cl> 1.446 CH3 CH3ntry> H 2(CH2)2try>CH-
NHCH3 H Cl
|
> 1.447 CH3 CH3ntry> H 0(CH2)2try>CH-
NHC2H5 H Cl
> 1.448 CH3 CH3ub>
H 2(CH2)2b>
CH-
NHC2H5 H Cl
> 1.449 CH3 CH3ub>
H 0(CH2)2b>
CH-
N(CH3)2 H Cl
> 1.450 CH3 CH3ub>
H 2(CH2)2b>
CH-
N(CH3)2 H Cl
> 1.451 CH3 CH3ub>
H 0(CH2)2b>
CH-
NHOC2H5 H Cl
w> 1.452 CH3 CH3<
/sub> H 2(CH2)2ub>
CH-
NHOC2H5 H Cl
w> 1.453 CH3 CH3<
/sub> H 0(CH2)2ub>
CH-
N(CH3)OC2H5 Hy> Cl
|
1.454 CH3ntry> CH3 H 2(CH
2)2CH-
N(CH3)OC2H5 Hy> Cl
1.455 CH3ntry> CH3 H 0(CH
2)2C＝N-
NH2 H Cl
1
.456 CH3 CH3y> H 2(CH2)2>C＝N-
NH2 H Cl 1
.457 CH3 CH3y> H 0(CH2)2>C＝N-
N(CH3)2 H Cl
> 1.458 CH3 CH3ub>
H 2(CH2)2b>
C＝N-
N(CH3)2 H Cl
> 1.459 CH3 CH3ub>
H 0(CH2)2b>
C(CH3)-
OCH3 H Cl
1.460 CH3 CH3ry> H 2(CH2)2y>C(CH3)-
OCH3 H Cl
1.461 CH3 CH3ry> H 0(CH2)2y>O H Cl 1.462
CH3 CH3 H
2(CH2)2O<
entry> H Cl 1.463 C>2H5
H H 0
>(CH2)2CH-
NHCH3 H Cl> 1.464 C2H5 Htry> H 2(CH2)2y>CH-
NHCH3 H Cl
|
> 1.465 C2H5 Htry> H 0(CH2)2y>CH-
NHC2H5 H Cl
> 1.466 C2H5
H H 2(CH2)2>
CH-
NHC2H5 H Cl
> 1.467 C2H5
H H 0(CH2)2>
CH-
N(CH3)2 H Cl
> 1.468 C2H5
H H 2(CH2)2>
CH-
N(CH3)2 H Cl
> 1.469 C2H5
H H 0(CH2)2>
CH-
NHOC2H5 H Cl
w> 1.470 C2H5> H H 2(CH2)2b>
CH-
NHOC2H5 H Cl
w> 1.471 C2H5> H H 0(CH2)2b>
CH-
N(CH3)OC2H5 Hy> Cl
1.472 C2H5ub>
H H 2(CH2
)2CH-
N(CH3)OC2H5 Hy> Cl
1.473 C2H5ub>
H H 0(CH2
)2C＝N-
NH2 H Cl
|
p>
olspec> 序号R15 R16 R<sup>17
n X Y L M
1.474> C2H5 H H
2(CH2)2 C＝N-
NH2 H Cl
1.475
C2H5 H H
0(CH2)2 C＝N-
N(CH3)2
H Cl> 1.476 C2H5
H H 2(CH2)2>
C＝N-
N(CH3)2 H Cl
> 1.477 C2H5
H H 0(CH2)2>
C(CH3)-
OCH3 H Cl
1.478
C2H5 Hy> H 2(CH2)2> C(CH3)-
OCH3 H Cl
1.479
C2H5 Hy> H 0(CH2)2> O H Cl
1.480 C2H5 H H<
entry> 2(CH2)2 Ontry> H Cl
1.481 CHb>3
CH3 H 0y>(CH2)2 CH-
NHCH3
CH3 CH3b>
1.482 CH3y> CH3 H 2(CH2sub>)2
CH-
NHCH3 CH3 CH3b>
1.483 CH3y> CH3 H 0(CH2sub>)2
CH-
NHC2H5 CH3
CH3
1.484 CH3>
CH3 H 2>(CH2)2 CH-
NHC2H5 CH3
CH3
1.485 CH3>
CH3 H 0>(CH2)2 CH-
N(CH3)2 CH3
CH3
1.486 CH3>
CH3 H 2>(CH2)2 CH-
N(CH3)2 CH3
CH3
1.487 CH3>
CH3 H 0>(CH2)2 CH-
NHOC2H5 CH3
CH3
1.488 CH3b>
CH3 H 2y>(CH2)2 CH-
NHOC2H5 CH3
CH3
1.489 CH3b>
CH3 H 0y>(CH2)2 CH-
N(CH3)OC2H5 CH3>
CH3
1.490> CH3 CH3 H> 2(CH2)2 CH-
N(CH3)OC2H5 CH3>
CH3
1.491> CH3 CH3 H> 0(CH2)2 C＝N-
NH2 CH3 CH3
1.492 CH3 CH3
H 2(CH2b>)2
C＝N-NH2
CH3 CH3
1.493 CH3 CH3
H 0(CH2b>)2
C＝N-N(CH3)2
CH3 CH3
1.494 CH3>
CH3 H 2>(CH2)2 C＝N-
N(CH3)2 CH3
CH3
1.495 CH3>
CH3 H 0>(CH2)2 C(CH3)-
OCH3 CH3 CH3>
1.496 CH3> CH3 H 2(CH2ub>)2
C(CH3)-
OCH3 CH3 CH3>
1.497 CH3> CH3 H 0(CH2ub>)2
O CH3> CH3
1.498 CH3ub>
CH3 H 2ry>(CH2)2 O CH3b>
CH3
1.499y> C2H5 H H> 0(CH2)2 CH-
NHCH3 CH3 CH3b>
1.500 C2H5>
H H 2(CH2ub>)2
CH-NHCH3
CH3 CH3b>
1.501 C2H5>
H H 0(CH2ub>)2
CH-NHC2H5
CH3 CH3
1.502 C2H5
H H 2(CH2)2
CH-NHC2H5
CH3 CH3
1.503 C2H5
H H 0(CH2)2
CH-N(CH3)2
CH3 CH3
1.504 C2H5
H H 2(CH2)2
CH-N(CH3)2
CH3 CH3
1.505 C2H5
H H 0(CH2)2
CH-NHOC2H5
CH3 CH3
1.506 C2H5
H H 2(CH2)2
CH-NHOC2H5
CH3 CH3
1.507 C2H5
H H 0(CH2)2
CH-N(CH3)OC2H5
CH3>
CH3
1.508> C2H5 H H
2(CH2)2 CH-
N(CH3)OC2H5 CH3>
CH3
1.509> C2H5 H H
0(CH2)2 C＝N-
NH CH3 CH3
> 1.510 C2H5
H H 2(CH2)2>
C＝N-
NH2 CH3 CH3
> 序号
R15 R16 R<
sup>17 n X Y L
M
1.511> C2H5 H H
0(CH2)2C＝N-
N(CH3)2 CH3
CH3
1.512 C2H5
H H 2(CH2)2
C＝N-N(CH3)2
CH3 CH3
1.513 C2H5
H H 0(CH2)2
C(CH3)-OCH3
CH3 CH3>
1.514 C2H5 H H 2(CH2b>)2
C(CH3)-OCH3
CH3 CH3>
1.515 C2H5 H H 0(CH2b>)2
O CH3 CH3
1.516 C2H5
H H 2(CH2)2
O CH3entry> CH3
1.517 CH3
CH3 H 0(CH2)2CH-NHCH3
Cl Cl
y> 1.518 CH3 CH3
H 2(CH2)2<
entry>CH-
NHCH3 Cl Cl
|
y> 1.519 CH3 CH3
H 0(CH2)2<
entry>CH-
NHC2H5 Cl Cl
> 1.520 CH3 CH3ub>
H 2(CH2)2b>
CH-
NHC2H5 Cl Cl
> 1.521 CH3 CH3ub>
H 0(CH2)2b>
CH-
N(CH3)2 Cl Cl
> 1.522 CH3 CH3ub>
H 2(CH2)2b>
CH-
N(CH3)2 Cl Cl
> 1.523 CH3 CH3ub>
H 0(CH2)2b>
CH-
NHOC2H5 Cl Cl
w> 1.524 CH3 CH3<
/sub> H 2(CH2)2ub>
CH-
NHOC2H5 Cl Cl
w> 1.525 CH3 CH3<
/sub> H 0(CH2)2ub>
CH-
N(CH3)OC2H5 Cly> Cl
|
1.526 CH3ntry> CH3 H 2(CH
2)2CH-
N(CH3)OC2H5 Cly> Cl
1.527 CH3ntry> CH3 H 0(CH
2)2C＝N-
NH2 Cl Cl
1.528
CH3 CH3ry> H 2(CH2)2y>C＝N-
NH2 Cl Cl
1.529
CH3 CH3ry> H 0(CH2)2y>C＝N-
N(CH3)2 Cl Cl
> 1.530 CH3 CH3ub>
H 2(CH2)2b>
C＝N-
N(CH3)2 Cl Cl
> 1.531 CH3 CH3ub>
H 0(CH2)2b>
C(CH3)-
OCH3 Cl Cl
1.532
CH3 CH3try> H 2(CH2)2y>C(CH3)-
OCH3 Cl Cl
|
1.533
CH3 CH3try> H 0(CH2)2y>O Cl Cl
|
1.534 CH3 CH3 H
2(CH2)2O<
entry> Cl Cl
1.535 Cb>2H5
H H 0y>(CH2)2CH-
NHCH3
Cl Cl
y> 1.536 C2H5 Hntry> H 2(CH2)2try>CH-
NHCH3 Cl Cl
|
y> 1.537 C2H5 Hntry> H 0(CH2)2try>CH-
NHC2H5 Cl Cl
> 1.538 C2H5
H H 2(CH2)2>
CH-
NHC2H5 Cl Cl
> 1.539 C2H5
H H 0(CH2)2>
CH-
N(CH3)2 Cl Cl
> 1.540 C2H5
H H 2(CH2)2>
CH-
N(CH3)2 Cl Cl
> 1.541 C2H5
H H 0(CH2)2>
CH-
NHOC2H5 Cl Cl
w> 1.542 C2H5> H H 2(CH2)2b>
CH-
NHOC2H5 Cl Cl
w> 1.543 C2H5> H H 0(CH2)2b>
CH-
N(CH3)OC2H5 Cly> Cl
1.544 C2H5ub>
H H 2(CH2
)2CH-
N(CH3)OC2H5 Cly> Cl
1.545 C2H5ub>
H H 0(CH2
)2C＝N-
NH2 Cl Cl
|
1.546
C2H5 H> H 2(CH2)2
C＝N-
NH2 Cl Cl
1.547
C2H5 H> H 0(CH2)2
C＝N-
N(CH3)2 Cl Cl
>
spec>> 序号
R15 R16 R
17 n X Y
L M
|
1.548y> C2H5 H H> 2(CH2)2C＝N-
N(CH3)2 Cl Cl
> 1.549 C2H5
H H 0(CH2)2>
C(CH3)-
OCH3 Cl Cl
1.550
C2H5 Hy> H 2(CH2)2>C(CH3)-
OCH3 Cl Cl
|
1.551
C2H5 Hy> H 0(CH2)2>O Cl Cl
|
1.552 C2H5 H H<
entry> 2(CH2)2Ontry> Cl Cl
1.553 CHb>3
CH3 H 0y>(CH2)2C＝
O
Cl Cl
1.554ntry> CH3 CH3 Hntry> 2(CH2)2C＝
O Cl Cl
1.555ntry> CH3 CH3 Hntry> 0(CH2)2CHOCH
3 Cl Cl
1.556try> CH3 CH3 Htry> 2(CH2)2CHOC
H3
Cl Cl
1.557
CH3 CH3> H 0(CH2)2
CHOC2H5 Cl Cl
w> 1.558 CH3 CH3<
/sub> H 2(CH2)2ub>
CHOC2H5 Clntry> Cl
1.559 CH3 CH3 H 0(CH>2)2
CHOiPr Cl Cl
1.560 CH3 CH3
H 2(CH2b>)2
CHOiPr Cl Cl>
1.561 CH3 CHb>3
H 0(CH2)>2
CHOH Cl Cl
<row> 1.562 CH3 CH3>
H 2(CH2)2
CHOH Cl Cltry> 1.563 CH3 CH3> H 0(CH2)2
C＝
NOCH3
Cl Cl
|
y> 1.564 CH3CH3<
entry> H 2(CH2)2ntry>C＝
NOCH3 Cl Cl
|
y> 1.565 CH3 CH3
H 0(CH2)2<
entry>C＝
NOC2H5 Cl Cl
> 1.566 CH3 CH3ub>
H 2(CH2)2b>
C＝
NOC2H5 Cl Cl
> 1.567 CH3 CH3ub>
H 0(CH2)2b>
C＝
NOiPr Cl Cl
|
1.568y> CH3 CH3 Hy> 2(CH2)2C＝
NOiPr
Cl Cl
1.569y> CH3 CH3 Hy> 0(CH2)2C＝
NOCH2CH＝
CHCl
Cl Cl
1.570> CH3 CH3 H> 2(CH2)2C＝
NOCH2CH＝
CHCl
Cl Cl
1.571> CH3 CH3 H> 0(CH2)2C＝
NOCH2C6H5
Cl> Cl
1.572 CH3try> CH3 H 2(CH2
)2C＝
NOCH2C6H5 Cl> Cl
1.573 CH3try> CH3 H 0(CH2
)2C(CH3)2y> Cl Cl
1.574 CH
3 CH3 H 2
(CH2)2C(CH3)2sub>
Cl Cl 1.575> C2H5 H H
0(CH2)2C＝
O
Cl Cl
1.576ntry> C2H5 H Hry> 2(CH2)2C＝
O Cl Cl
1.577ntry> C2H5 H Hry> 0(CH2)2CHOCH3
Cl Cl
1.578y> C2H5 H H> 2(CH2)2CHOCHub>3
Cl Cl
1.579
C2H5 H Hentry> 0(CH2)2CHO
C2H5
Cl Cl<
row> 1.580 C2H5 H
H 2(CH2)2<
/entry>CHOC2H5 Cl
Cl 1.581 C2H5
H H 0(CH2b>)2
CHOiPr ClCl> 1.582 C2H5
H H 2(CH2)>2
CHOiPr Cl Cl
1.583 C2H5
H
H 0(CH2)2>
CHOH Cl Clntry> 1.584 C2H5 H
H 2(CH2)2<
entry>CHOH Cl Cl
|
</table>ec> 序号 R15 R16 R<sup>17
n X Y L M
1.585> C2H5 H H
0(CH2)2C＝
NOCH3 Cl Cl
y> 1.586 C2H5 Hntry> H 2(CH2)2try>C＝
NOCH3 Cl Cl
|
y> 1.587 C2H5 Hntry> H 0(CH2)2try>C＝
NOC2H5 Cl Cl
> 1.588 C2H5
H H 2(CH2)2>
C＝
NOC2H5 Cl Cl
> 1.589 C2H5
H H 0(CH2)2>
C＝
NOiPr Cl Cl
|
1.590y> C2H5 H H> 2(CH2)2C＝
NOiPr
Cl Cl
1.591y> C2H5 H H> 0(CH2)2C＝
NOCH2CH＝
CHCl
Cl Cl
1.592> C2H5 H H
2(CH2)2C＝
NOCH2CH＝
CHCl
Cl Cl
1.593> C2H5 H H
0(CH2)2C＝
NOCH2C6H5
Cl> Cl
1.594 C2H5b>
H H 2(CH2sub>)2
C＝NOCH2C6H5
Cl> Cl
1.595 C2H5b>
H H 0(CH2sub>)2
C(CH3)2 Cl
Cl
1.596 C2ub>H5
H H 2ry>(CH2)2C(CH3)2>
Cl Cl
1.597ntry> CH3 CH3 Hntry> 0(CH2)2C＝
O CH3 CH3
<row> 1.598 CH3 CH3>
H 2(CH2)2
C＝
O CH3 CH3<
row> 1.599 CH3 CH3>
H 0(CH2)2
CHOCH3 CH3y> CH3 1.600 CH3sub>
CH3 H 2ntry>(CH2)2CHOCH3<
entry> CH3 CH3
> 1.601 CH3 CH3ntry> H 0(CH2)2try>CHOC2H5 CH3try> CH3
|
1.602 CH3
CH3 H 2<
entry>(CH2)2CHOC2H5<
/sub> CH3 CH3
w> 1.603 CH3 CH3<
/sub> H 0(CH2)2ub>
CHOiPr CH3 CH>3
1.604 CH3> CH3 H 2(CHub>2)2
CHOiPr CH3entry> CH3
1.605 C
H3 CH3 H 0
(CH2)2CHOH> CH3 CH3 1.
606 CH3 CH3> H 2(CH2)2
CHOH CH3 CH3
ow> 1.607 CH3 CH3
H 0(CH2)2<
/sub>C＝
NOCH3 CH3 CH3b>
1.608 CH3y> CH3 H 2(CH2sub>)2
C＝
NOCH3 CH3 CH3b>
1.609 CH3y> CH3 H 0(CH2sub>)2
C＝
NOC2H5 CH3
CH3
1.610 CH3>
CH3 H 2>(CH2)2C＝
NOC2H5 CH3
CH3
1.611 CH3>
CH3 H 0>(CH2)2C＝
NOiPr CH3 CH3
w> 1.612 CH3 CH3<
/sub> H 2(CH2)2ub>
C＝
NOiPr CH3 CH3
w> 1.613 CH3 CH3<
/sub> H 0(CH2)2ub>
C＝NOCH2CH＝
CHCl CH3 CH3
w> 1.614 CH3 CH3<
/sub> H 2(CH2)2ub>
C＝NOCH2CH＝
CHCl CH3 CH3
w> 1.615 CH3 CH3<
/sub> H 0(CH2)2ub>
C＝
NOCH2C6H5 CH3
CH3
1.616
CH3 CH3 H
2(CH2)2C＝
NOCH2C6H5 CH3
CH3 1.617
CH3 CH3 H
0(CH2)2C(CH3
)2 CH3 CH3ntry> 1.618 CH3 C
H3
H 2(CH2
)2C(CH3)2 CH<
sub>3 CH3 1.619ntry> C2H5 H Hry> 0(CH2)2C＝
O
CH3 CH3
<
row> 1.620 C2H5 H
H 2(CH2)2<
/entry>C＝
O CH3 CH3<
row> 1.621 C2H5 H
H 0(CH2)2<
/entry>CHOCH3 CH3> CH3
c> 序号 R15 R16 R17
n X Y L
M
1.622y> C2H5 H H> 2(CH2)2CHOCH3sub>
CH3 CH3
> 1.623 C2H5
H H 0(CH2)2>
CHOC2H5 CH3>
CH3
1.624> C2H5 H H
2(CH2)2CHOC2>H5
CH3 CH3<
/entry>
1.625 C2H5ntry> H H 0(CH2)
2
CHOiPr CH3> CH3
1.626 C2>H5
H H 2>(CH2)2CHOiPr CH3
CH3
1.627<entry> C2H5 H Hntry> 0(CH2)2CHOH> CH3 CH3
try> 1.628 C2H5 H<
entry> H 2(CH2)2ntry>CHOH CH3 CH3y>
|
1.629 C2H5> H H 0(CH2)b>2
C＝
NOCH3
CH3 CH3b>
1.630 C2H5>
H H 2(CH2ub>)2
C＝NOCH3
CH3 CH3b>
1.631 C2H5>
H H 0(CH2ub>)2
C＝NOC2H5
CH3 CH3
1.632 C2H5
H H 2(CH2)2
C＝NOC2H5
CH3 CH3
1.633 C2H5
H H 0(CH2)2
C＝NOiPr
CH3 CH3w> 1.634 C2H5> H H 2(CH2)2b>
C＝
NOiPr CH3 CH3
w> 1.635 C2H5> H H 0(CH2)2b>
C＝NOCH2CH＝
CHCl CH3 CH3
w> 1.636 C2H5> H H 2(CH2)2b>
C＝NOCH2CH＝
CHCl CH3 CH3
w> 1.637 C2H5> H H 0(CH2)2b>
C＝
NOCH2C6H5 CH3
CH3
1.638
C2H5 H H 2
(CH2)2C＝
NOCH2C6H5 CH3
CH3
1.639
C2H5 H H 0
(CH2)2C(CH3)
2 CH3 CH3try>
1.640 C2H5y> H H 2(CH2)ub>2
C(CH3)2 CHb>3
CH3
表2：下式化合物
<colspec> 序号R15 R16 R<sup>17
n X Y L M
2.1 CH3
CH3 H 0
N COCH3 Hntry> CH3
2.2 CH3 CH3 H 2<entry> N COCH3 H CHub>3
2.3 CH3y> CH3 H 0 Nntry> COC2H5 H CH
3
2.4 CH3ntry> CH3 H 2 N<
/entry> COC2H5 H C
H3
2.5 CH3</entry> CH3 H 0
N
COiPr H CH3</row> 2.6 CH3 CH3
H 2 N COiPrentry> H CH3
2.7</entry> C2H5 H Hntry> 0 N COCH3
H
CH3
2.8> C2H5 H H
2 N COCH3 Hntry> CH3
2.9 C2ub>H5
H H 0ry> N COC2H5 Hntry> CH3
2.10 C2</sub>H5
H H 2ntry> N COC2H5 H
CH3
2.11 C2
H5 H H 0 N COiPr H CH3<
/entry>
2.12 C2H5ntry> H H 2 N
COiPr
H CH3
> 2.13 CH3 CH3ntry> H 0 CH COCH3
ntry> H CH3
|
2.14 CH3 CH3 H 2 CH COCH3ntry> H CH3
2.15 CH3 CH3 H
0 CH COC2H5y> H CH3
2.16ntry> CH3 CH3 Hntry> 2 CH COC2H5
H CH3
2.17
CH3 CH3 H
0 CH COiPr Hry> CH3
2.18 CH<sub>3
CH3 H 2ntry> CH COiPr H CH3<
/sub>
2.19 C2H5ub>
H H 0 CH COCH3 H CH3ry>
2.20 C2H5> H H 2 CH C
OCH3
H CH3> 2.21 C2H5
H H 0 CH COC2
H5 H CH3
ow> 2.22 C2H5y> H H 2 CH COCb>2H5
H CH3>
2.23 C2H5
H H 0 CH CO
iPr H CH3
2.24
C2H5 H> H 2 CH COiPr Hntry> CH3
2.25 CH3
CH3 H 0 N COCH3 Hry> Cl
2.26 CH3<entry> CH3 H 2 N> COCH3 H Cl
w> 2.27 CH3 CH3<
/entry> H 0 N COC2b>H5
H Cl
2.28 CH3 CH3ry> H 2 N COC2H5
H Cl 2.29y> CH3 CH3 Hy> 0 N COiPr H> Cl
ec>ead> 序号
R15 R16 R
17 n X Y
L M
2.30> CH3 CH3 H> 2 NCOiPr H Cly>
2.31 C2H5 H H 0 NCOC
H3 H Cl
2.32
C2H5 H H
2 NCOCH3try> H Cl
2.33 C2H5 H H 0<entry> NCOC2H5 H
Cl
2.34 C2H5
H H 2 Ny>COC2H5 H Cltry>
2.35 C2H5> H H 0 NCOi
Pr
H Cl
2.36try> C2H5 H Hy> 2 NCOiPr H Cl
try>
2.37 CH3 CH<sub>3
H 0 CHCOCH3
H Cl
2.38
CH3 CH3y> H 2 CHCOCH3> H Cl
2.39 CH<sub>3
CH3 H 0ntry> CHCOC2H5 H
Cl
2.40 CH3>
CH3 H 2> CHCOC2H5 Htry> Cl
2.41 CH3ntry> CH3 H 0 CH>COiPr H Cl
2.42
CH3 CH3 H
2 CHCOiPr Hy> Cl
2.43 C2Hb>5
H H 0 CH</entry>COCH3 H Cl
> 2.44 C2H5
H
H 2 CHCOCH3
H Cl
2.45y> C2H5 H H> 0 CHCOC2H5ry> H Cl
2.46 C2H5
H H 2entry> CHCOC2H5
H
Cl
2.47 C2>H5
H H 0> CHCOiPr H Cl
2.48 C2H5 H> H 2 CHCOiPr> H
Cl
|
表3：下式
化合物
<colspec> 序号R15 R16 R<sup>17
n Y L M
3.1 CH3>
CH3 H 0> COCH3 H CH3
ow> 3.2 CH3 CH3<
/sub> H 2 COCH3
> H CH3
3.3y> CH3 CH3 Hy> 0 COC2H5 Hry> CH3
3.4 CHub>3
CH3 H 2try> COC2H5 H CH<
sub>3
3.5 CH3ry> CH3 H 0 COi
Pr
H CH3
3.6
CH3 CH3> H 2 COiPr H CHb>3
3.7 C2H5
H H 0 COCH3
H CH3
w> 3.8 C2H5 Hntry> H 2 COCH3
H
CH3 3.9> C2H5 H H
0 COC2H5 H> CH3
3.10 C2>H5
H H 2> COC2H5 H CH3b>
3.11 C2H5>
H H 0 COiPr> H CH3
3.12ry> C2H5 H H> 2 COiPr H CH3
3.13 CH3
CH3 H 0 COCH3sub>
H Cl 3.14
CH3 CH3 H
2 COCH3 H Clentry> 3.15 CH3 C
H3
H 0 COC2>H5
H Cl
3.16 CH3 CH3y> H 2 COC2H5ry> H Cl 3.17 CH>3
CH3 H 0> COiPr H Cl
3
.18 CH3 CH3> H 2 COiPr H Cl
ry> 3.19 C2H5> H H 0 COCH3<
/entry> H Cl
3.20y> C2H5 H H> 2 COCH3 H Cl
3.21 C2H5ntry> H H 0 COC2H>5
H Cl
3.22ntry> C2H5 H Hry> 2 COC2H5 Hntry> Cl
3.23 C2H
5 H H 0 C
OiPr H Cl 3.24
C2H5 H H<
entry> 2 COiPr H Cl
body>
表4：下式化合物
<colspec> 序号 R15 R16 R<sup>17
n X Y M
L
4.1> CH3 CH3 H> 0 CH2C＝
O H CH3
4.2
CH3 CH3 H
2 CH2C＝O
H CH3
4.3
CH3 CH3 H
0 CH2CHOCH3</sub>
H CH3
> 4.4 CH3 CH3ry> H 2 CH2CHOCH>3
H CH3
|
ntry> 4.5 CH3 CH3
H 0 CH2CHOC<
sub>2H5 H CH3y>
|
4.6 CH3 CH>3
H 2 CH2>CHOC2H5 H CHub>3
4.7 CH3> CH3 H 0 CHb>2
CHOiPr H CH3
4.8 CH3 CH3
H 2 CH2CHOiPr H CH3row> 4.9 CH3 CH3sub>
H 0 CH2ntry>CHOH H CH3
|
4.10 CH3 CH3ry> H 2 CH2CHO
H
H CH3
4.11
CH3 CH3 H
0 CH2C＝NOCH3
H CH3w> 4.12 CH3 CH3sub>
H 2 CH2ntry>C＝
NOCH3 H CH3
w> 4.13 CH3 CH3sub>
H 0 CH2ntry>C＝
NOC2H5 H CH3>
4.14 CH3
CH3 H 2 CH2>
C＝
NOC2H5 H CH3>
4.15 CH3
CH3 H 0 CH2>
C＝
NOiPr H CH3
y> 4.16 CH3 CH3ntry> H 2 CH2C＝
NOiPr H CH3
|
y> 4.17 CH3 CH3ntry> H 0 CH2C＝
NOCH2CH＝
CHCl H CH3
|
> 4.18 CH3 CH3try> H2 CH2C＝
NOCH2CH＝
CHCl H CH3
|
> 4.19 CH3 CH3try> H 0 CH2C＝
NOCH2C6H5 H
CH3
|
4.20 CH3>
CH3 H 2> CH2C＝
NOCH2C6H5 H
CH3
4.21 CH3>
CH3 H 0> CH2C(CH3)2
H CH3
4.22 CH3
CH3 H 2
CH2C(CH3)2 H CH3
4.23
C2H5 H H 0 CH2C＝O
H CH3
4.24
C2H5 H H
2 CH2C＝O
H CH3
4.25
C2H5 H H
0 CH2CHOCH3</sub>
H CH3
> 4.26 C2H5 Hy> H 2 CH2CHOCH>3
H CH3
|
ntry> 4.27 C2H5 H<
entry> H 0 CH2CHOCb>2H5
H CH3>
|
4.28 C2H5<entry> H H 2 CH2>CHOC2H5 H CHub>3
4.29 C2H>5
H H 0 CHub>2
CHOiPr H CH3>
>d> 序号
R15 R16R<
sup>17 n X Y
M L
4.30> C2H5 H H
2 CH2CHOiPr H
CH3
4.31 C2H5 H H 0<entry> CH2CHOH H CH
3
4.32 C2Hb>5
H H 2 CH<sub>2
CHOH H CH3>
4.33 C2H5entry> H H 0 CH2
C＝NOCH3
H CH3w> 4.34 C2H5
H H 2 CH2y>C＝
NOCH3 H CH3
w> 4.35 C2H5
H H 0 CH2y>C＝
NOC2H5 H CH3>
4.36 C2H5entry> H H 2 CH2
C＝NOC2H5
H CH3>
4.37 C2H5entry> H H 0 CH2
C＝NOiPr
H CH3
y> 4.38 C2H5 Htry> H 2 CH2C＝
NOiPr H CH3
|
y> 4.39 C2H5 Htry> H 0 CH2C＝
NOCH2CH＝
CHCl H CH3
|
> 4.40 C2H5 Hy> H 2 CH2C＝
NOCH2CH＝
CHCl H CH3
|
> 4.41 C2H5 Hy> H 0 CH2C＝
NOCH2C6H5 H
CH3
|
4.42 C2H5
H H 2 CH2
C＝NOCH2C6H5
H CH3
4.43 C2H5
H H 0 CH2
C(CH3)2 H
CH3
4.44 C2H5
H H 2 CH2C(CH3)2entry> H CH3
4.45</entry> CH3 CH3 H<
/entry> 0 CH2C＝
O
H Cl
4.46ry> CH3 CH3 Hry> 2 CH2C＝
O H Cl
4.47ry> CH3 CH3 Hry> 0 CH2CHOCH3
H Cl
4.48 CHub>3
CH3 H 2try> CH2CHOCH3 H
Cl
4.49 CH3>
CH3 H 0> CH2CHOC2H5> H Cl
4.50 CH3</sub>
CH3 H 2ntry> CH2CHOC2H5ntry> H Cl
4.51 CH>3
CH3 H 0> CH2CHOiPr H
Cl
4.52 CH3> CH3 H 2 CH2ub>
CHOiPr H Cl
> 4.53 CH3 CH3try> H 0 CH2CH
OH
H Cl 4.54ntry> CH3 CH3 Hntry> 2 CH2CHOH Htry> Cl
4.55 CH3ntry> CH3 H 0 C
H2
C＝
NOCH3 H Cl> 4.56 CH3 CH3try> H 2 CH2C＝
NOCH3 H Cl
|
> 4.57 CH3 CH3try> H 0 CH2C＝
NOC2H5 H Cl
|
> 4.58 CH3 CH3b>
H 2 CH2y>C＝
NOC2H5 H Cl
> 4.59 CH3 CH3b>
H 0 CH2y>C＝
NOiPr H Cl
4.60> CH3 CH3 H> 2 CH2C＝
NOiPr
H Cl
4.61> CH3 CH3 H> 0 CH2C＝
NOCH2CH＝
CHCl
H Cl
4.62
CH3 CH3 H
2 CH2C＝
NOCH2CH＝
CHCl H Cl
4.63
CH3 CH3 H
0 CH2C＝
NOCH2C6H5 H
Cl 4.64 CH3> CH3 H 2 CH2ub>
C＝
NOCH2C6H5 H
Cl
4.65 CH3> CH3 H 0 CH2ub>
C(CH3)2 Hy> Cl
4.66 CH3try> CH3 H 2 CH2<
/sub>C(CH3)2 Htry> Cl
lspec>
序号 R15 R16 R17
n X Y M
L
4.67y> C2H5 H H> 0 CH2C＝
O H Cl
4.68ntry> C2H5 H Hry> 2 CH2C＝
O H Cl
4.69ntry> C2H5 H Hry> 0 CH2CHOCH3
H Cl
4.70 Cub>2H5
H H 2try> CH2CHOCH3 H
Cl
4.71 C2>H5
H H 0> CH2CHOC2H5> H Cl
4.72 C2sub>H5
H H 2ntry> CH2CHOC2H5ntry> H Cl
4.73 C>2H5
H H 0> CH2CHOiPr H
Cl
4.74 C2H5 H H 2 CH2b>
CHOiPr H Cl
4.75 C2H5 Hy> H 0 CH2CHO
H
H Cl
|
4.76ntry> C2H5 H Hry> 2 CH2CHOH Hy> Cl
4.77 C2Hub>5
H H 0 CH2
C＝NOCH3
H Cl
> 4.78 C2H5 Htry> H 2 CH2C＝
NOCH3 H Cl
|
> 4.79 C2H5 Htry> H 0 CH2C＝
NOC2H5 H Cl
> 4.80 C2H5
H H 2 CH2>C＝
NOC2H5 H Cl
> 4.81 C2H5
H H 0 CH2>C＝
NOiPr H Cl
|
4.82> C2H5 H H
2 CH2C＝
NOiPr
H Cl
4.83> C2H5 H H
0 CH2C＝
NOCH2CH＝
CHCl
H Cl
4.84> C2H5 H H
2 CH2C＝
NOCH2CH＝
CHCl
H Cl
4.85> C2H5 H H
0 CH2C＝
NOCH2C6H5
H Cl
4.86 C2H5>
H H 2 CH2ub>
C＝NOCH2C6H5
H Cl
4.87 C2H5>
H H 0 CH2ub>
C(CH3)2 Hy> Cl
4.88 C2H5ub>
H H 2 CH2C(CH3)2 Hntry> Cl
4.89 CH3 CH3 H 0(CH>2)2
C＝
O H Cl
4.90ntry> CH3 CH3 Hntry> 2(CH2)2C＝
O H Cl
4.91ntry> CH3 CH3 Hntry> 0(CH2)2CHOCH
3 H Cl
4.92ry> CH3 CH3 Hry> 2(CH2)2CHOCH
3
H Cl
4.93
CH3 CH3 H
0(CH2)2CHOC2H5
H Cl> 4.94 CH3 CH3ub>
H 2(CH2)2b>
CHOC2H5 Hry> Cl
4.95 CH3<
entry> CH3 H 0(CH
2)2CHOiPr H Clentry>
4.96 CH3 CH3
H 2(CH2)2
CHOiPr H Clrow> 4.97 CH3 CH
3 H 0(CH2)2
CHOH H Cl
w> 4.98 CH3 CH3<
/entry> H 2(CH2)2entry>CHOH H Cl> 4.99
|
CH3 CH3ntry> H 0(CH2)2try>C＝
NOCH3 H Cl> 4.100 CH3 CH3
H 2(CH2)2<
entry>C＝
NOCH3 H Cl
|
> 4.101 CH3 CH3
H 0(CH2)2<
entry>C＝
NOC2H5 H Cl
> 4.102 CH3 CH3sub>
H 2(CH2)2ub>
C＝
NOC2H5 H Cl
> 4.103 CH3 CH3sub>
H 0(CH2)2ub>
C＝
NOiPr H Cl
|
olspec> 序号R15 R16 R<sup>17
n X Y M
L
4.104y> CH3 CH3 Hy> 2(CH2)2C＝
NOiPr H Cl
4.105> CH3 CH3 H> 0(CH2)2C＝
NOCH2CH＝
CHCl
H Cl
4.106> CH3 CH3 H> 2(CH2)2C＝
NOCH2CH＝
CHCl
H Cl
4.107> CH3 CH3 H> 0(CH2)2C＝
NOCH2C6H5
H
Cl
4.108 CH3y> CH3 H 2(CH2sub>)2
C＝
NOCH2C6H5 H
Cl
4.109 CH3y> CH3 H 0(CH2sub>)2
C(CH3)2
H Cl
4.110 CH3sub>
CH3 H 2ntry>(CH2)2C(CH3)2b>
H Cl
4.111<entry> C2H5 H Hntry> 0(CH2)2C＝
O H Cl
4.112ntry> C2H5 H Hry> 2(CH2)2C＝
O H Cl
4.113ntry> C2H5 H Hry> 0(CH2)2CHOCH3
H Cl
4.114y> C2H5 H H> 2(CH2)2CHOCHub>3
H Cl
4.115</entry> C2H5 H Hntry> 0(CH2)2CHOC
2H5
H Cl
w> 4.116 C2H5 Hentry> H 2(CH2)2ntry>CHOC2H5 H Cl
4.117 C2H5entry> H H 0(CH2
)2
CHOiPr H Clrow> 4.118 C2H5ry> H
H 2(CH2)2sub>
CHOiPr H Cl> 4.119 C2H5 Htry> H 0(CH2)2y>CHOH H Cl 4
.120
C2H5 H
H
2(CH2)2C
HOH H Cl 4.121> C2H5 H H
0(CH2)2C＝
NOCH3
H Cl
> 4.122 C2H5 Htry> H 2(CH2)2y>C＝
NOCH3 H Cl
|
> 4.123 C2H5 Htry> H 0(CH2)2y>C＝
NOC2H5 H Cl
|
> 4.124 C2H5
H H 2(CH2)2>
C＝
NOC2H5 H Cl
> 4.125 C2H5
H H 0(CH2)2>
C＝
NOiPr H Cl 4.126> C2H5 H H
2(CH2)2C＝
NOiPr
H Cl
4.127> C2H5 H H
0(CH2)2C＝
NOCH2CH＝
CHCl
H Cl
4.128> C2H5 H H
2(CH2)2C＝
NOCH2CH＝
CHCl
H Cl
4.129> C2H5 H H
0(CH2)2C＝
NOCH2C6H5
H
Cl 4.130 C2H5>
H H 2(CH2ub>)2
C＝
NOCH2C6H5 H
Cl 4.131 C2H5>
H H 0(CH2ub>)2
C(CH3)2
H Cl 4.132 C2b>H5
H H 2y>(CH2)2C(CH3)2
H Cl
4.133ry> CH3 CH3 Hry> 0(CH2)2C＝
O H CH3
4.
134 CH3 CH3> H 2(CH2)2
C＝
O H CH3 4.
135 CH3 CH3> H 0(CH2)2
CHOCH3 H CH3
ow> 4.136 CH3 CH3
H 2(CH2)2<
/sub>CHOCH3 H CHb>3
4.137 CH3y> CH3 H 0(CH<
sub>2)2
CHOC2H5y> H CH3
4.138ntry> CH3 CH3 Hntry> 2(CH2)2CHOC
2H5
H CH3try>
4.139 CH3 CH
3 H 0(CH2)<
sub>2CHOiPr H CH3b>
4.140 CH3y> CH3 H 2(CH2sub>)2
CHOiPr H CH>3
<colspec>c> 序号R15 R16Rup>17
n X Y M L
4.141> CH3 CH3 H> 0(CH2)2CHOHntry> H CH3
4.142 CH3 CH3 H
2(CH2)2CHOHry> H CH3
4.143ntry> CH3 CH3 Hntry> 0(CH2)2C＝
NOCH3
H CH3
w> 4.144 CH3 CH3<
/sub>
H 2(CH2)2ub>
C＝NOCH3
H CH3w> 4.145 CH3 CH3<
/sub> H 0(CH2)2ub>
C＝
NOC2H5 H CH3>
4.146 CH3> CH3 H 2(CH2ub>)2
C＝
NOC2H5 H CH3>
4.147 CH3> CH3 H 0(CH2ub>)2
C＝
NOiPr H CH3
y> 4.148 CH3 CH3
H 2(CH2)2<
entry>C＝
NOiPr H CH3
|
y> 4.149 CH3 CH3
H 0(CH2)2<
entry>C＝NOCH2CH＝
CHCl H CH3
|
> 4.150 CH3 CH3ntry> H 2(CH2)2try>C＝NOCH2CH＝
CHCl H CH3
|
> 4.151 CH3 CH3ntry> H 0(CH2)2try>C＝
NOCH2C6H5 H
CH3
|
4.152 CH3b>
CH3 H 2y>(CH2)2C＝
NOCH2C6H5 H
CH3
4.153 CH3b>
CH3 H 0y>(CH2)2C(CH3)2
H CH3
4.154
CH3 CH3 H
2(CH2)2C(CH3)2
H CH3</entry>
4.155 C2H5ntry> H H 0(CH2)
2
C＝O
H CH3
4.156
C2H5 H H
2(CH2)2C＝
O
H CH3
4.157
C2H5 H H
0(CH2)2CHOCH3
H CH3w> 4.158 C2H5> H H 2(CH2)2b>
CHOCH3 H CH3
4.159 C2H5sub>
H H 0(CH2
)2CHOC2H5ry> H CH3
4.160ntry> C2H5 H Hry> 2(CH2)2CHOC2sub>H5
H CH3
w> 4.161 C2H5> H H 0(CH2)2b>
CHOiPr H CH3
>
4.162 C2H5
H H 2(CH2)>2
CHOiPr H CH3
4.163 C2H5entry> H H 0(CH2
)2
CHOH H CH3ub>
4.164 C2H5>
H H 2(CH2ub>)2
CHOH H CH3
4.165 C2H5 H H 0(CH>2)2
C＝NOCH3
H CH3w> 4.166 C2H5> H H 2(CH2)2b>
C＝
NOCH3 H CH3
w> 4.167 C2H5> H H 0(CH2)2b>
C＝
NOC2H5 H CH3>
4.168 C2H5
H H 2(CH2b>)2
C＝
NOC2H5 H CH3>
4.169 C2H5
H H 0(CH2b>)2
C＝
NOiPr H CH3
y> 4.170 C2H5 Hntry> H 2(CH2)2try>C＝
NOiPr H CH3
|
y> 4.171 C2H5 Hntry> H 0(CH2)2try>C＝NOCH2CH＝
CHCl H CH3
|
> 4.172 C2H5 Htry> H 2(CH2)2y>C＝NOCH2CH＝
CHCl H CH3
|
> 4.173 C2H5 Htry> H 0(CH2)2y>C＝
NOCH2C6H5 H
CH3
|
4.174 C2H5
H H 2(CH2)2
C＝NOCH2C6H5
H CH3
4.175 C2H5
H H 0(CH2)2
C(CH3)2ntry> H CH3
4.176 C2H5 H Hentry> 2(CH2)2C(CH
3)2
H CH3ry>
4.177 CH3 CH<sub>3
p-CH3-C6H4-SO2-
0(CH2)2C＝
O
H CH3
>
lspec> 序号R15 R16 R<sup>17
nX Y M L
4.178> CH3 CH3 p-
CH3-C6H4-SO2-
2(CH2)2C＝
O H CH3
4.179
CH3 CH3> p-CH3-C6H4-SO2-
0(CH2)2CH
OCH3 H CH3
> 4.180 CH3 CH3ub>
p-CH3-C6H4-
SO2-
2(CH2)2CH
OCH3 H CH3
> 4.181 CH3 CH3ub>
P-CH3-C6H4-
SO2-
0(CH2)2CH
OC2H5 H CH3
4.182 CH3 CH3
p-CH3-C6H4-SO2-
2(CH2)2CHOC2H5
H CH3
4.183 CH3 CH3
p-CH3-C6H4-SO2-
0(CH2)2CHOiPr
H CH3
4.184
CH3 CH3try> p-CH3-C6H4-SO2-
2(CH2)2CH
OiPr H CH3
|
4.185
CH3 CH3try> p-CH3-C6H4-SO2-
0(CH2)2CH
OH H CH3
|
4.186
CH3 CH3ry> p-CH3-C6H4-SO2-
2(CH2)2CH
OH H CH3
4.187
CH3 CH3ry> p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH3 H CH3
w> 4.188 CH3 CH3<
/sub> p-CH3-C6H4-
SO2-
2(CH2)2C＝
NOCH3 H CH3
w> 4.189 CH3 CH3<
/sub> p-CH3-C6H4-
SO2-
0(CH2)2C＝
NOC2H5 H CH3>
4.190 CH3> CH3 p-CH3-
C6H4-SO2-
2(CH2)2C＝
NOC2H5 H CH3>
4.191 CH3> CH3 p-CH3-
C6H4-SO2-
0(CH2)2C＝
NOiPr H CH3
y> 4.192 CH3 CH3
p-CH3-C6H4-SO2-
2(CH2)2C＝
NOiPr H CH3
|
y> 4.193 CH3 CH3
p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH2CH＝
CHCl H CH3
|
> 4.194 CH3 CH3ntry> P-CH3-C6H4-SC2-
2(CH2)2C＝
NOCH2CH＝
CHCl H CH3
|
> 4.195 CH3 CH3ntry> p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH2C6H5 H
CH3
|
4.196 CH3b>
CH3 p-CH3-C6H4-SO2-
2(CH2)2C＝NOCH2C6H5
H CH3
4.197 CH3b>
CH3 p-CH3-C6H4-SO2-
0(CH2)2C(CH3)2
H CH3ntry>
4.198 CH3 CH3
P-CH3-C6H4-SO2-
2(CH2)2C(CH3)2
H CH3ntry>
4.199 C2H5ry> H p-CH3-C6H4-
SO2-
0(CH2)2C＝O
H CH3
4.200
C2H5 H p-CH3-C6H4-SO2-
2(CH2)2C＝O
H CH3
4.201
C2H5 H P-CH3-C6H4-SO2-
0(CH2)2CHOCH3
H CH3> 4.202 C2H5
H P-CH3-C6H4-
SO2-
2(CH2)2CH
OCH3 H CH3
> 4.203 C2H5
H p-CH3-C6H4-
SO2-
0(CH2)2CH
OC2H5 H CH3
4.204 C2H5entry> H p-CH3-C6H4-
SO2-
2(CH2)2CHOC2H5
H CH3
4.205 C2H5entry> H p-CH3-C6H4-
SO2-
0(CH2)2CHOiPr
H CH3
4.206
C2H5 Hy> P-CH3-C6H4-SO2-
2(CH2)2CH
OiPr H CH3
|
4.207
C2H5 Hy> P-CH3-C6H4-SO2-
0(CH2)2CH
OH H CH3
|
4.208
C2H5 H> p-CH3-C6H4-SO2-
2(CH2)2CH
OH H CH3
4.209
C2H5 H> p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH3 H CH3
w> 4.210 C2H5> H p-CH3-C6H4-
SO2-
2(CH2)2C＝
NOCH3 H CH3
w> 4.211 C2H5> H p-CH3-C6H4-
SO2-
0(CH2)2C＝
NOC2H5 H CH3>
4.212 C2H5
H p-CH3-
C6H4-SO2-
2(CH2)2C＝
NOC2H5 H CH3>
4.213 C2H5
H P-CH3-
C6H4-SO2-
0(CH2)2C＝
NOiPr H CH3
y> 4.214 C2H5 Hntry> p-CH3-C6H4-SO2-
2(CH2)2C＝
NOiPr H CH3
|
group>
c> 序号R15R16 Rup>17
n X Y M L
4.215> C2H5 H p-
CH3-C6H4-SO2-
0(CH2)2 C
＝NOCH2CH＝
CHCl H CH3
> 4.216 C2H5 Htry> p-CH3-C6H4-SO2-
2(CH2)2 C
＝NOCH2CH＝
CHCl H CH3
|
> 4.217 C2H5 Htry> p-CH3-C6H4-SO2-
0(CH2)2 C
＝
NOCH2C6H5 H
CH3
|
4.218 C2H5
H p-CH3-C6H4-SO2-
2(CH2)2 C＝
NOCH2C6H5
H CH3
4.219 C2H5
H p-CH3-C6H4-SO2-
0(CH2)2 C(CH3)2
H CH3entry>
4.220 C2H5try> H p-CH3-C6H4-
SO2-
2(CH2)2 C(CH3)2
H CH3entry>
4.221 CH3 CH3
H0(CH2)2
CH-NHCH3
H CH3w> 4.222 CH3 CH3<
/sub> H2(CH2)2ub>
CH-
NHCH3 H CH3
w> 4.223 CH3 CH3<
/sub> H0(CH2)2ub>
CH-
NHC2H5 H CH3>
4.224 CH3> CH3 H2(CH2b>)2
CH-
NHC2H5 H CH3>
4.225 CH3> CH3 H0(CH2b>)2
CH-
N(CH3)2 H CH3>
4.226 CH3> CH3 H2(CH2b>)2
CH-
N(CH3)2 H CH3>
4.227 CH3> CH3 H0(CH2b>)2
CH-
NHOC2H5 H CH3b>
4.228 CH3y> CH3 H2(CH2ub>)2
CH-
NHOC2H5 H CH3b>
4.229 CH3y> CH3 H0(CH2ub>)2
CH-
N(CH3)OC2H5 Hy> CH3
4.230 CH3sub>
CH3 H2try>(CH2)2 CH-
N(CH3)OC2H5 Hy> CH3
4.231 CH3sub>
CH3 H0try>(CH2)2 C＝N-
NH2 H CH3
<row> 4.232 CH3 CH3>
H2(CH2)2
C＝N-
NH2 H CH3<
row> 4.233 CH3 CH3>
H0(CH2)2
C＝N-
N(CH3)2 H CH3>
4.234 CH3> CH3 H2(CH2b>)2
C＝N-
N(CH3)2 H CH3>
4.235 CH3> CH3 H0(CH2b>)2
C(CH3)-
OCH3 H CH3
> 4.236 CH3 CH3ub>
H2(CH2)2b>
C(CH3)-
OCH3 H CH3
> 4.237 CH3 CH3ub>
H0(CH2)2b>
O H CH3w> 4.238 CH3 CH3<
/sub> H2(CH2)2ub>
O H CH3
ow> 4.239 C2H5y> H H0(CH2)2ub>
CH-
NHCH3 H CH3
w> 4.240 C2H5> H H2(CH2)2b>
CH-
NHCH3 H CH3
w> 4.241 C2H5> H H0(CH2)2b>
CH-
NHC2H5 H CH3>
4.242 C2H5
H H2(CH2>)2
CH-
NHC2H5 H CH3>
4.243 C2H5
H H0(CH2>)2
CH-
N(CH3)2 H CH3>
4.244 C2H5<
/entry> H H2(CH2
)2 CH-
N(CH3)2 H CH3>
4.245 C2H5
H H0(CH2>)2
CH-
NHOC2H5 H CH3b>
4.246 C2H5>
H H2(CH2ub>)2
CH-
NHOC2H5 H CH3b>
4.247 C2H5>
H H0(CH2ub>)2
CH-
N(CH3)OC2H5 Hy> CH3 4.248 C2b>H5
H H2y>(CH2)2 CH-
N(CH3)OC2H5 Hy> CH3
4.249 C2b>H5
H H0y>(CH2)2 C＝N-
NH2 H CH3
<
row> 4.250 C2H5 H
H2(CH2)2entry> C＝N-
NH2
H CH3<
row> 4.251 C2H5 H
H0(CH2)2entry> C＝N-
N(CH3)2
H CH3>
>d> 序号
R15 R16 R<
sup>17 n X Y
M L
4.252y> C2H5 H H> 2(CH2)2 C＝N-
N(CH3)2 H CH3>
4.253 C2H5 H H 0(CH2b>)2
C(CH3)-OCH3
H CH3> 4.254 C2H5
H H 2(CH2)2>
C(CH3)-
OCH3 H CH3
> 4.255 C2H5
H H 0(CH2)2>
O H CH3
> 4.256 C2H5
H H 2(CH2)2>
O H CH3
> 4.257 CH3 CH3ub>
H 0(CH2)2b>
CH-
NHCH3 H Cl
> 4.258 CH3 CH3ntry> H 2(CH2)2try> CH-
NHCH3 H Cl
|
> 4.259 CH3 CH3ntry> H 0(CH2)5try> CH-
NHC2H5 H Cl
> 4.260 CH3 CH3ub>
H 2(CH2)2b>
CH-
2024年5月7日发(作者：冷书文)
2(CH2)2C＝
NOiPr H Cl
|
1.171> C2H5 H H
0(CH2)2C＝
NOCH2CH＝
CHCl
H Cl
1.172> C2H5 H H
2(CH2)2C＝
NOCH2CH＝
CHCl
H Cl
1.173> C2H5 H H
0(CH2)2C＝
NOCH2C6H5
H Cl
1.174 C2H5>
H H 2(CH2ub>)2
C＝NOCH2C6H5
H Cl
1.175 C2H5>
H H 0(CH2ub>)2
C(CH3)2 H
Cl
1.176 C2b>H5
H H 2y>(CH2)2C(CH3)2
H Cl
1.177ry> CH3 CH3 Hry> 0(CH2)2C＝
O H CH3
>
lspec> 序号 R15 R16 R<sup>17
n X Y L M
1.178> CH3 CH3 H> 2(CH2)2C＝
O H CH3
1.179
CH3 CH3> H 0(CH2)2
CHOCH3 H CH3
ow> 1.180 CH3 CH3
H 2(CH2)2<
/sub>CHOCH3 H CHb>3
1.181 CH3y> CH3 H 0(CH<
sub>2)2
CHOC2H5y> H CH3
1.182ntry> CH3 CH3 Hntry> 2(CH2)2CHOC
2H5
H CH3try>
1.183 CH3 CH3
H 0(CH2)<sub>2
CHOiPr H CH3b>
1.184 CH3y> CH3 H 2(CH2sub>)2
CHOiPr H CH>3
1.185 CH3> CH3 H 0(CHub>2)2
CHOH H C
H3
1.186 CH3 CH3 H 2(CH2)2
CHOH Htry> CH3
1.187 CH3 CH3 H 0<entry>(CH2)2C＝
NOCH3 H CH3
w> 1.188 CH3 CH3<
/sub> H 2(CH2)2ub>
C＝
NOCH3 H CH3
w> 1.189 CH3 CH3<
/sub> H 0(CH2)2ub>
C＝
NOC2H5 H CH3>
1.190 CH3> CH3 H 2(CH2ub>)2
C＝
NOC2H5 H CH3>
1.191 CH3> CH3 H 0(CH2ub>)2
C＝
NOiPr H CH3
y> 1.192 CH3 CH3
H 2(CH2)2<
entry>C＝
NOiPr H CH3
|
y> 1.193 CH3 CH3
H 0(CH2)2<
entry>C＝NOCH2CH＝
CHCl H CH3
|
> 1.194 CH3 CH3ntry> H 2(CH2)2try>C＝NOCH2CH＝
CHCl H CH3
|
> 1.195 CH3 CH3ntry> H 0(CH2)2try>C＝
NOCH2C6H5 H
CH3
|
1.196 CH3b>
CH3 H 2y>(CH2)2C＝
NOCH2C6H5 H
CH3
1.197 CH3b>
CH3 H 0y>(CH2)2C(CH3)2
H CH3
1.198
CH3 CH3 H
2(CH2)2C(CH3)2
H CH3</entry>
1.199 C2H5ntry> H H 0(CH2)
2
C＝O
H CH3
1.200
C2H5 H H
2(CH2)2C＝
O
H CH3
1.201
C2H5 H H
0(CH2)2CHOCH3
H CH3w> 1.202 C2H5> H H 2(CH2)2b>
CHOCH3 H CH3
1.203 C2H5sub>
H H 0(CH2
)2CHOC2H5ry> H CH3
1.204ntry> C2H5 H Hry> 2(CH2)2CHOC2sub>H5
H CH3
w> 1.205 C2H5> H H 0(CH2)2b>
CHOiPr H CH3
>
1.206 C2H5
H H 2(CH2)>2
CHOiPr H CH3
1.207 C2H5entry> H H 0(CH2
)2
CHOH H CH3ub>
1.208 C2H5>
H H 2(CH2ub>)2
CHOH H CH3
1.209 C2H5 H H 0(CH>2)2
C＝NOCH3
H CH3w> 1.210 C2H5> H H 2(CH2)2b>
C＝
NOCH3 H CH3
w> 1.211 C2H5> H H 0(CH2)2b>
C＝
NOC2H5 H CH3>
1.212 C2H5
H H 2(CH2b>)2
C＝
NOC2H5 H CH3>
1.213 C2H5
H H 0(CH2b>)2
C＝
NOiPr H CH3
y> 1.214 C2H5 Hntry> H 2(CH2)2try>C＝
NOiPr H CH3
|
group>
c> 序号 R15 R16 R<sup>17
n X Y L M
1.215> C2H5 H H
0(CH2)2C＝
NOCH2CH＝
CHCl H CH3
> 1.216 C2H5 Htry> H2(CH2)2y>C＝NOCH2CH＝
CHCl H CH3
|
> 1.217 C2H5 Htry> H0(CH2)2y>C＝
NOCH2C6H5 H
CH3
|
1.218 C2H5
H H2(CH2)2
C＝NOCH2C6H5
H CH3
1.219 C2H5
H H0(CH2)2
C(CH3)2ntry> H CH3
1.220 C2H5 H Hentry>2(CH2)2C(CH
3)2
H CH3ry>
1.221 CH3 CH<sub>3
p-CH3-C6H4-SO2-
0(CH2)2C＝O
H CH3
1.222
CH3 CH3> p-CH3-C6H4-SO2-
2(CH2)2C＝
O H CH3
1.223
CH3 CH3> p-CH3-C6H4-SO2-
0(CH2)2CH
OCH3 H CH3
> 1.224 CH3 CH3ub>
p-CH3-C6H4-
SO2-
2(CH2)2CH
OCH3 H CH3
> 1.225 CH3 CH3ub>
p-CH3-C6H4-
SO2-
0(CH2)2CH
OC2H5 H CH3
1.226 CH3 CH3
p-CH3-C6H4-SO2-
2(CH2)2CHOC2H5
H CH3
1.227 CH3 CH3
P-CH3-C6H4-SO2-
0(CH2)2CHOiPr
H CH3
1.228
CH3 CH3try> p-CH3-C6H4-SO2-
2(CH2)2CH
OiPr H CH3
|
1.229
CH3 CH3try> p-CH3-C6H4-SO2-
0(CH2)2CH
OH H CH3
|
1.230
CH3 CH3ry> P-CH3-C6H4-SC2-
2(CH2)2CH
OH H CH3
1.231
CH3 CH3ry> p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH3 H CH3
w> 1.232 CH3 CH3<
/sub> p-CH3-C6H4-
SO2-
2(CH2)2C＝
NOCH3 H CH3
w> 1.233 CH3 CH3<
/sub> p-CH3-C6H4-
SO2-
0(CH2)2C＝
NOC2H5 H CH3>
1.234 CH3> CH3 p-CH3-
C6H4-SO2-
2(CH2)2C＝
NOC2H5 H CH3>
1.235 CH3> CH3 p-CH3-
C6H4-SO2-
0(CH2)2C＝
NOiPr H CH3
y> 1.236 CH3 CH3
p-CH3-C6H4-SO2-
2(CH2)2C＝
NOiPr H CH3
|
y> 1.237 CH3 CH3
p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH2CH＝
CHCl H CH3
|
> 1.238 CH3 CH3ntry> p-CH3-C6H4-SO2-
2(CH2)2C＝
NOCH2CH＝
CHCl H CH3
|
> 1.239 CH3 CH3ntry> p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH2C6H5 H
CH3
|
1.240 CH3b>
CH3 p-CH3-C6H4-SO2-
2(CH2)2C＝NOCH2C6H5
H CH3
1.241 CH3b>
CH3 p-CH3-C6H4-SO2-
0(CH2)2C(CH3)2
H CH3ntry>
1.242 CH3 CH3
p-CH3-C6H4-SO2-
2(CH2)2C(CH3)2
H CH3ntry>
1.243 C2H5ry> H p-CH3-C6H4-
SO2-
0(CH2)2C＝O
H CH3
1.244
C2H5 H p-CH3-C6H4-SO2-
2(CH2)2C＝O
H CH3
1.245
C2H5 H p-CH3-C6H4-SO2-
0(CH2)2CHOCH3
H CH3> 1.246 C2H5
H p-CH3-C6H4-
SO2-
2(CH2)2CH
OCH3 H CH3
> 1.247 C2H5
H p-CH3-C6H4-
SC2-
0(CH2)2CH
OC2H5 H CH3
1.248 C2H5entry> H p-CH3-C6H4-
SO2-
2(CH2)2CHOC2H5
H CH3
1.249 C2H5entry> H p-CH3-C6H4-
SO2-
0(CH2)2CHOiPr
H CH3
1.250
C2H5 Hy> p-CH3-C6H4-SO2-
2(CH2)2CH
OiPr H CH3
|
1.251
C2H5 Hy> p-CH3-C6H4-SO2-
0(CH2)2CH
OH H CH3
|
up>
<colspec> 序号R15 R16 R<sup>17
n X Y L M
1.252> C2H5 H p-
CH3-C6H4-SO2-
2(CH2)2CH
OH H CH3
1.253
C2H5 H> p-CH3-C6H4-SO2-
0(CH2)2C
＝
NOCH3 H CH3
w> 1.254 C2H5> H p-CH3-C6H4-
SO2-
2(CH2)2C
＝
NOCH3 H CH3
w> 1.255 C2H5> H p-CH3-C6H4-
SO2-
0(CH2)2C
＝
NOC2H5 H CH3>
1.256 C2H5
H p-CH3-
C6H4-SO2-
2(CH2)2C
＝
NOC2H5 H CH3>
1.257 C2H5
H p-CH3-
C6H4-SO2-
0(CH2)2C
＝
NOiPr H CH3
y> 1.258 C2H5 Hntry> p-CH3-C6H4-SO2-
2(CH2)2C
＝
NOiPr H CH3
|
y> 1.259 C2H5 Hntry> p-CH3-C6H4-SO2-
0(CH2)2C
＝NOCH2CH＝
CHCl H CH3
|
> 1.260 C2H5 Htry> p-CH3-C6H4-SO2-
2(CH2)2C
＝NOCH2CH＝
CHCl H CH3
|
> 1.261 C2H5 Htry> p-CH3-C6H4-SO2-
0(CH2)2C
＝
NOCH2C6H5 H
CH3
|
1.262 C2H5
H p-CH3-C6H4-SO2-
2(CH2)2C＝
NOCH2C6H5
H CH3
1.263 C2H5
H p-CH3-C6H4-SO2-
0(CH2)2C(CH3)2
H CH3entry>
1.264 C2H5try> H P-CH3-C6H4-
SO2-
2(CH2)2C(CH3)2
H CH3entry>
1.265 CH3 CH3
H 0 CH2CH-NHCH3
H H
> 1.266 CH3 CH3ntry> H 2 CH2CH-
NHCH3 H H
|
> 1.267 CH3 CH3ntry> H 0 CH2CH-
NHC2H5 H H
> 1.268 CH3 CH3ub>
H 2 CH2ry>CH-
NHC2H5 H H
> 1.269 CH3 CH3ub>
H 0 CH2ry>CH-
N(CH3)2 H H
> 1.270 CH3 CH3ub>
H 2 CH2ry>CH-
N(CH3)2 H H
> 1.271 CH3 CH3ub>
H 0 CH2ry>CH-
NHOC2H5 H H
w> 1.272 CH3 CH3<
/sub> H 2 CH2ntry>CH-
NHOC2H5 H H
w> 1.273 CH3 CH3<
/sub> H 0 CH2ntry>CH-
N(CH3)OC2H5 Hy> H
1.274 CH3ntry> CH3 H 2 CH2
CH-
N(CH3)OC2H5 Hy> H
1.275 CH3ntry> CH3 H 0 CH2
C＝N-
NH2 H H
1
.276 CH3 CH3y> H 2 CH2C＝N-
NH2 H H
1
.277 CH3 CH3y> H 0 CH2C＝N-
N(CH3)2 H H
> 1.278 CH3 CH3ub>
H 2 CH2ry>C＝N-
N(CH3)2 H H
> 1.279 CH3 CH3ub>
H 0 CH2ry>C(CH3)-
OCH3 H H
1.280 CH3 CH3ry> H 2 CH2C(CH3
)-
OCH3 H H
1.281 CH3 CH3ry> H 0 CH2Ontry> H H
1.282 CHb>3
CH3 H 2y> CH2O H H
ntry>
|
1.283 C2H5ry> H H 0 CH2ntry>CH-
NHCH3
H H
> 1.284 C2H5 Htry> H 2 CH2CH-
NHCH3 H H
|
> 1.285 C2H5 Htry> H 0 CH2CH-
NHC2H5 H H
> 1.286 C2H5
H H 2 CH2>CH-
NHC2H5 H H
> 1.287 C2H5
H H 0 CH2>CH-
N(CH3)2 H H
> 1.288 C2H5
H H 2 CH2>CH-
N(CH3)2 H H
>
|
spec>> 序号
R15 R16 R<
sup>17 n X Y L
M
|
1.289> C2H5 H H
0 CH2 CH-
NHOC2H5 H H
w> 1.290 C2H5> H H 2 CH2ry> CH-
NHOC2H5 H H
w> 1.291 C2H5> H H 0 CH2ry> CH-
N(CH3)OC2H5 Hy> H
1.292 C2H5b>
H H 2 CH2sub>
CH-
N(CH3)OC2H5 Hy> H
1.293 C2H5b>
H H 0 CH2sub>
C＝N-
NH2 H H
1.294
C2H5 H H
2 CH2 C＝N-NH2
H H
1.295
C2H5 H H
0 CH2 C＝N-N(CH3)2
H H> 1.296 C2H5
H H 2 CH2> C＝N-
N(CH3)2 H H
> 1.297 C2H5
H H 0 CH2> C(CH3)-
OCH3 H H
1.298
C2H5 H> H 2 CH2 C(CH3<
/sub>)-
OCH3 H H
1.299
C2H5 H> H 0 CH2 Ory> H H
1.300 C2H5 H H 2<entry> CH2 O H H>
1.301 CH3 CHb>3
H 0 CH2y> CH-
NHCH3
H CH3w> 1.302 CH3 CH3<
/sub> H 2 CH2ntry> CH-
NHCH3 H CH3
w> 1.303 CH3 CH3<
/sub> H 0 CH2ntry> CH-
NHC2H5 H CH3>
1.304 CH3> CH3 H 2 CH2ub>
CH-
NHC2H5 H CH3>
1.305 CH3> CH3 H 0 CH2ub>
CH-
N(CH3)2 H CH3>
1.306 CH3> CH3 H 2 CH2ub>
CH-
N(CH3)2 H CH3>
1.307 CH3> CH3 H 0 CH2ub>
CH-
NHOC2H5 H CH3b>
1.308 CH3y> CH3 H 2 CH2sub>
CH-
NHOC2H5 H CH3b>
1.309 CH3y> CH3 H 0 CH2sub>
CH-
N(CH3)OC2H5 Hy> CH3
1.310 CH3sub>
CH3 H 2ntry> CH2 CH-
N(CH3)OC2H5 Hy> CH3
1.311 CH3sub>
CH3 H 0ntry> CH2 C＝N-
NH2 H CH3
<row> 1.312 CH3 CH3>
H 2 CH2> C＝N-
NH2 H CH3<
row> 1.313 CH3 CH3>
H 0 CH2> C＝N-
N(CH3)2 H CH3>
1.314 CH3> CH3 H 2 CH2ub>
C＝N-
N(CH3)2 H CH3>
1.315 CH3> CH3 H 0 CH2ub>
C(CH3)-
OCH3 H CH3
> 1.316 CH3 CH3ub>
H 2 CH2ry> C(CH3)-
OCH3 H CH3
> 1.317 CH3 CH3ub>
H 0 CH2ry> O H CH3
> 1.318 CH3 CH3ntry> H 2 CH2 O
H CH3
|
1.319y> C2H5 H H
> 0 CH2 CH-
NHCH3 H CH3
w> 1.320 C2H5> H H 2 CH2ry> CH-
NHCH3 H CH3
w> 1.321 C2H5> H H 0 CH2ry> CH-
NHC2H5 H CH3>
1.322 C2H5
H H 2 CH2b>
CH-
NHC2H5 H CH3>
1.323 C2H5
H H 0 CH2b>
CH-
N(CH3)2 H CH3>
1.324 C2H5
H H 2 CH2b>
CH-
N(CH3)2 H CH3>
1.325 C2H5
H H 0 CH2b>
CH-
NHOC2H5 H CH3b>
c>ad> 序号
R15 R16 R<
sup>17 n X Y L
M
1.326> C2H5 H H
2 CH2 CH-
NHOC2H5 H CH3b>
1.327 C2H5>
H H 0 CH2ub>
CH-N(CH3)OC2H5
Hy> CH3
1.328 C2b>H5
H H 2y> CH2 CH-
N(CH3)OC2H5 Hy> CH3
1.329 C2b>H5
H H 0y> CH2 C＝N-
NH2 H CH3
<row> 1.330 C2H5 H
H2 CH2
C＝N-
NH2 H CH3<
row> 1.331 C2H5 H
H 0 CH2
C＝N-
N(CH3)2 H CH3>
1.332 C2H5
H H 2 CH2b>
C＝N-
N(CH3)2 H CH3>
1.333 C2H5
H H 0 CH2b>
C(CH3)-
OCH3 H CH3
> 1.334 C2H5
H H 2 CH2> C(CH3)-
OCH3 H CH3
> 1.335 C2H5
H H 0 CH2> O H CH3
1.336 C2H5 Hy> H 2 CH2 Ontry> H CH3 1.337
CH3 CH3 H
0 CH2 CH-
NHCH3 H Cl> 1.338 CH3 CH3ntry> H 2 CH2 CH-
NHCH3 H Cl
|
> 1.339 CH3 CH3ntry> H 0 CH2 CH-
NHC2H5 H Cl
> 1.340 CH3 CH3ub>
H 2 CH2ry> CH-
NHC2H5 H Cl
> 1.341 CH3 CH3ub>
H 0 CH2ry> CH-
N(CH3)2 H Cl
> 1.342 CH3 CH3ub>
H 2 CH2ry> CH-
N(CH3)2 H Cl
> 1.343 CH3 CH3ub>
H 0 CH2ry> CH-
NHOC2H5 H Cl
w> 1.344 CH3 CH3<
/sub> H 2 CH2ntry> CH-
NHOC2H5 H Cl
w> 1.345 CH3 CH3<
/sub> H 0 CH2ntry> CH-
N(CH3)OC2H5 Hy> Cl
1.346 CH3ntry> CH3 H 2 CH2
CH-
N(CH3)OC2H5 Hy> Cl
1.347 CH3ntry> CH3 H 0 CH2
C＝N-
NH2 H Cl
1
.348 CH3 CH3y> H 2 CH2 C＝N-
NH2 H Cl
1
.349 CH3 CH3y> H 0 CH2 C＝N-
N(CH3)2 H Cl
> 1.350 CH3 CH3ub>
H 2 CH2ry> C＝N-
N(CH3)2 H Cl
> 1.351 CH3 CH3ub>
H 0 CH2ry> C(CH3)-
OCH3 H Cl
1.352 CH3 CH3ry> H 2 CH2 C(CH
3)-
OCH3 H Cl
1.353 CH3 CH3ry> H 0 CH2 Ontry> H Cl
1.354 CHb>3
CH3 H 2
|
y> CH2 O H Clentry> 1.355 C2H5try> H H 0 CH2entry> CH-
NHCH3
H Cl
> 1.356
|
C2H5 Htry> H 2 CH2 CH-
NHCH3 H Cl> 1.357 C2H5 Htry> H 0 CH2 CH-
NHC2H5 H Cl
> 1.358 C2H5
H H 2 CH2> CH-
NHC2H5 H Cl
> 1.359 C2H5
H H 0 CH2> CH-
N(CH3)2 H Cl
> 1.360 C2H5
H H 2 CH2> CH-
N(CH3)2 H Cl
> 1.361 C2H5
H H 0 CH2> CH-
NHOC2H5 H Cl
w> 1.362 C2H5> H H 2 CH2ry> CH-
NHOC2H5 H Cl
w>
|
olspec>y> 序号
R15 R16 R<
sup>17 n X Y L
M
|
1.363> C2H5 H H
0 CH2 CH-
N(CH3)OC2H5 Hy> Cl
1.364 C2H5ub>
H H 2 CH2 CH-N(CH3)OC2H5
Hy> Cl
1.365 C2H5ub>
H H 0 CH2 C＝N-NH2
H Cl
1.366
C2H5 H H
2 CH2 C＝N-NH2
H Cl
1.367
C2H5 H H
0 CH2 C＝N-N(CH3)2
H Cl> 1.368 C2H5
H H 2 CH2> C＝N-
N(CH3)2 H Cl
> 1.369 C2H5
H H 0 CH2> C(CH3)-
OCH3 H Cl
1.370
C2H5 Hy> H 2 CH2 C(CH3
)-
OCH3 H Cl
1.371
C2H5 Hy> H 0 CH2 Ontry> H Cl
1.372 C>2H5
H H 2> CH2 O H Clntry>
1.373 CH3 CH3
H 0(CH2)2
CH-NHCH3
H H
> 1.374 CH3 CH3ntry> H 2(CH2)2try> CH-
NHCH3 H H
|
> 1.375 CH3 CH3ntry> H 0(CH2)2try> CH-
NHC2H5 H H
> 1.376 CH3 CH3ub>
H 2(CH2)2b>
CH-
NHC2H5 H H
> 1.377 CH3 CH3ub>
H 0(CH2)2b>
CH-
N(CH3)2 H H
> 1.378 CH3 CH3ub>
H 2(CH2)2b>
CH-
N(CH3)2 H H
> 1.379 CH3 CH3ub>
H 0(CH2)2b>
CH-
NHOC2H5 H H
w> 1.380 CH3 CH3<
/sub> H 2(CH2)2ub>
CH-
NHOC2H5 H H
w> 1.381 CH3 CH3<
/sub> H 0(CH2)2ub>
CH-
N(CH3)OC2H5 Hy> H
|
1.382 CH3ntry> CH3 H 2(CH
2)2 CH-
N(CH3)OC2H5 Hy> H
1.383 CH3ntry> CH3 H 0(CH
2)2 C＝N-
NH2 H H
1.384
CH3 CH3y> H 2(CH2)2> C＝N-
NH2 H H
1.385
CH3 CH3y> H 0(CH2)2> C＝N-
N(CH3)2 H H
> 1.386 CH3 CH3ub>
H 2(CH2)2b>
C＝N-
N(CH3)2 H H
> 1.387 CH3 CH3ub>
H 0(CH2)2b>
C(CH3)-
OCH3 H H
1.388
CH3 CH3ry> H 2(CH2)2y> C(CH3)-
OCH3 H H
1.389
CH3 CH3ry> H 0(CH2)2y> O H H
1.390 CH3 CH3 H
2(CH2)2 O<
entry> H H
1.391 C>2H5
H H 0>(CH2)2 CH-
NHCH3
H H
> 1.392 C2H5 Htry> H 2(CH2)2y> CH-
NHCH3 H H
|
> 1.393 C2H5 Htry> H 0(CH2)2y> CH-
NHC2H5 H H
> 1.394 C2H5
H H 2(CH2)2>
CH-
NHC2H5 H H
> 1.395 C2H5
H H 0(CH2)2>
CH-
N(CH3)2 H H
> 1.396 C2H5
H H 2(CH2)2>
CH-
N(CH3)2 H H
> 1.397 C2H5
H H 0(CH2)2>
CH-
NHOC2H5 H H
w> 1.398 C2H5> H H 2(CH2)2b>
CH-
NHOC2H5 H H
w> 1.399 C2H5> H H 0(CH2)2b>
CH-
N(CH3)OC2H5 Hy> H
|
pec>head> 序号
R15 R16 R<
sup>17 n XY L
M
1.400> C2H5 H H
2(CH2)2CH-
N(CH3)OC2H5 Hy> H
1.401 C2H5b>
H H 0(CH2sub>)2
C＝N-NH2
H H
1.402
C2H5 H H
2(CH2)2C＝N-
NH2
H H
1.403
C2H5 H H
0(CH2)2C＝N-
N(CH3)2
H H> 1.404 C2H5
H H 2(CH2)2>
C＝N-
N(CH3)2 H H
> 1.405 C2H5
H H 0(CH2)2>
C(CH3)-
OCH3 H H
1.406
C2H5 H> H 2(CH2)2
C(CH3)-
OCH3 H H
1.407
C2H5 H> H 0(CH2)2
O H H
1.408try> C2H5 H Hy> 2(CH2)2O> H H
1.409 CH3 CH3 H 0<entry>(CH2)2CH-
NHCH3 H CH3
w> 1.410 CH3 CH3> H 2(CH2)2
CH-
NHCH3
H CH3w> 1.411 CH3 CH3<
/sub> H 0(CH2)2ub>
CH-
NHC2H5 H CH3>
1.412 CH3> CH3 H 2(CH2ub>)2
CH-
NHC2H5 H CH3>
1.413 CH3> CH3 H 0(CH2ub>)2
CH-
N(CH3)2 H CH3>
1.414 CH3> CH3 H 2(CH2ub>)2
CH-
N(CH3)2 H CH3>
1.415 CH3> CH3 H 0(CH2ub>)2
CH-
NHOC2H5 H CH3b>
1.416 CH3y> CH3 H 2(CH2sub>)2
CH-
NHOC2H5 H CH3b>
1.417 CH3y> CH3 H 0(CH2sub>)2
CH-
N(CH3)OC2H5 Hy> CH3
1.418 CH3sub>
CH3 H 2ntry>(CH2)2CH-
N(CH3)OC2H5 Hy> CH3
1.419 CH3sub>
CH3 H 0ntry>(CH2)2C＝N-
NH2 H CH3
<
row> 1.420 CH3 CH3>
H 2(CH2)2
C＝N-
NH2 H CH3
<row> 1.421 CH3 CH3>
H 0(CH2)2
C＝N-
N(CH3)2 H CH3>
1.422 CH3> CH3 H 2(CH2ub>)2
C＝N-
N(CH3)2 H CH3>
1.423 CH3> CH3 H 0(CH2ub>)2
C(CH3)-
OCH3 H CH3
> 1.424 CH3 CH3ub>
H 2(CH2)2b>
C(CH3)-
OCH3 H CH3
> 1.425 CH3 CH3ub>
H 0(CH2)2b>
O H CH3> 1.426 CH3 CH3ub>
H 2(CH2)2b>
O H CH3> 1.427 C2H5
H H 0(CH2)2>
CH-
NHCH3 H CH3
w> 1.428 C2H5> H H 2(CH2)2b>
CH-
NHCH3 H CH3
w> 1.429 C2H5> H H 0(CH2)2b>
CH-
NHC2H5 H CH3>
1.430 C2H5
H H 2(CH2b>)2
CH-
NHC2H5 H CH3>
1.431 C2H5
H H 0(CH2b>)2
CH-
N(CH3)2 H CH3>
1.432 C2H5
H H 2(CH2b>)2
CH-
N(CH3)2 H CH3>
1.433 C2H5
H H 0(CH2b>)2
CH-
NHOC2H5 H CH3b>
1.434 C2H5>
H H 2(CH2ub>)2
CH-
NHOC2H5 H CH3b>
1.435 C2H5>
H H 0(CH2ub>)2
CH-
N(CH3)OC2H5 Hy> CH3 1.436 C2b>H5
H H 2y>(CH2)2CH-
N(CH3)OC2H5 Hy> CH3
>ec> 序号 R15 R16 R<sup>17
n XY L M
1.437> C2H5 H H
0(CH2)2C＝N-
NH2 H CH3
<row> 1.438 C2H5 H
H 2(CH2)2<
/entry>C＝N-
NH2 H CH3<
row> 1.439 C2H5 H
H 0(CH2)2<
/entry>C＝N-
N(CH3)2 H CH3>
1.440 C2H5
H H 2(CH2b>)2
C＝N-
N(CH3)2 H CH3>
1.441 C2H5
H H 0(CH2b>)2
C(CH3)-
OCH3 H CH3
> 1.442 C2H5
H H 2(CH2)2>
C(CH3)-
OCH3 H CH3
> 1.443 C2H5
H H 0(CH2)2>
O H CH3
> 1.444 C2H5
H H 2(CH2)2>
O H CH3
> 1.445 CH3 CH3ub>
H 0(CH2)2b>
CH-
NHCH3 H Cl> 1.446 CH3 CH3ntry> H 2(CH2)2try>CH-
NHCH3 H Cl
|
> 1.447 CH3 CH3ntry> H 0(CH2)2try>CH-
NHC2H5 H Cl
> 1.448 CH3 CH3ub>
H 2(CH2)2b>
CH-
NHC2H5 H Cl
> 1.449 CH3 CH3ub>
H 0(CH2)2b>
CH-
N(CH3)2 H Cl
> 1.450 CH3 CH3ub>
H 2(CH2)2b>
CH-
N(CH3)2 H Cl
> 1.451 CH3 CH3ub>
H 0(CH2)2b>
CH-
NHOC2H5 H Cl
w> 1.452 CH3 CH3<
/sub> H 2(CH2)2ub>
CH-
NHOC2H5 H Cl
w> 1.453 CH3 CH3<
/sub> H 0(CH2)2ub>
CH-
N(CH3)OC2H5 Hy> Cl
|
1.454 CH3ntry> CH3 H 2(CH
2)2CH-
N(CH3)OC2H5 Hy> Cl
1.455 CH3ntry> CH3 H 0(CH
2)2C＝N-
NH2 H Cl
1
.456 CH3 CH3y> H 2(CH2)2>C＝N-
NH2 H Cl 1
.457 CH3 CH3y> H 0(CH2)2>C＝N-
N(CH3)2 H Cl
> 1.458 CH3 CH3ub>
H 2(CH2)2b>
C＝N-
N(CH3)2 H Cl
> 1.459 CH3 CH3ub>
H 0(CH2)2b>
C(CH3)-
OCH3 H Cl
1.460 CH3 CH3ry> H 2(CH2)2y>C(CH3)-
OCH3 H Cl
1.461 CH3 CH3ry> H 0(CH2)2y>O H Cl 1.462
CH3 CH3 H
2(CH2)2O<
entry> H Cl 1.463 C>2H5
H H 0
>(CH2)2CH-
NHCH3 H Cl> 1.464 C2H5 Htry> H 2(CH2)2y>CH-
NHCH3 H Cl
|
> 1.465 C2H5 Htry> H 0(CH2)2y>CH-
NHC2H5 H Cl
> 1.466 C2H5
H H 2(CH2)2>
CH-
NHC2H5 H Cl
> 1.467 C2H5
H H 0(CH2)2>
CH-
N(CH3)2 H Cl
> 1.468 C2H5
H H 2(CH2)2>
CH-
N(CH3)2 H Cl
> 1.469 C2H5
H H 0(CH2)2>
CH-
NHOC2H5 H Cl
w> 1.470 C2H5> H H 2(CH2)2b>
CH-
NHOC2H5 H Cl
w> 1.471 C2H5> H H 0(CH2)2b>
CH-
N(CH3)OC2H5 Hy> Cl
1.472 C2H5ub>
H H 2(CH2
)2CH-
N(CH3)OC2H5 Hy> Cl
1.473 C2H5ub>
H H 0(CH2
)2C＝N-
NH2 H Cl
|
p>
olspec> 序号R15 R16 R<sup>17
n X Y L M
1.474> C2H5 H H
2(CH2)2 C＝N-
NH2 H Cl
1.475
C2H5 H H
0(CH2)2 C＝N-
N(CH3)2
H Cl> 1.476 C2H5
H H 2(CH2)2>
C＝N-
N(CH3)2 H Cl
> 1.477 C2H5
H H 0(CH2)2>
C(CH3)-
OCH3 H Cl
1.478
C2H5 Hy> H 2(CH2)2> C(CH3)-
OCH3 H Cl
1.479
C2H5 Hy> H 0(CH2)2> O H Cl
1.480 C2H5 H H<
entry> 2(CH2)2 Ontry> H Cl
1.481 CHb>3
CH3 H 0y>(CH2)2 CH-
NHCH3
CH3 CH3b>
1.482 CH3y> CH3 H 2(CH2sub>)2
CH-
NHCH3 CH3 CH3b>
1.483 CH3y> CH3 H 0(CH2sub>)2
CH-
NHC2H5 CH3
CH3
1.484 CH3>
CH3 H 2>(CH2)2 CH-
NHC2H5 CH3
CH3
1.485 CH3>
CH3 H 0>(CH2)2 CH-
N(CH3)2 CH3
CH3
1.486 CH3>
CH3 H 2>(CH2)2 CH-
N(CH3)2 CH3
CH3
1.487 CH3>
CH3 H 0>(CH2)2 CH-
NHOC2H5 CH3
CH3
1.488 CH3b>
CH3 H 2y>(CH2)2 CH-
NHOC2H5 CH3
CH3
1.489 CH3b>
CH3 H 0y>(CH2)2 CH-
N(CH3)OC2H5 CH3>
CH3
1.490> CH3 CH3 H> 2(CH2)2 CH-
N(CH3)OC2H5 CH3>
CH3
1.491> CH3 CH3 H> 0(CH2)2 C＝N-
NH2 CH3 CH3
1.492 CH3 CH3
H 2(CH2b>)2
C＝N-NH2
CH3 CH3
1.493 CH3 CH3
H 0(CH2b>)2
C＝N-N(CH3)2
CH3 CH3
1.494 CH3>
CH3 H 2>(CH2)2 C＝N-
N(CH3)2 CH3
CH3
1.495 CH3>
CH3 H 0>(CH2)2 C(CH3)-
OCH3 CH3 CH3>
1.496 CH3> CH3 H 2(CH2ub>)2
C(CH3)-
OCH3 CH3 CH3>
1.497 CH3> CH3 H 0(CH2ub>)2
O CH3> CH3
1.498 CH3ub>
CH3 H 2ry>(CH2)2 O CH3b>
CH3
1.499y> C2H5 H H> 0(CH2)2 CH-
NHCH3 CH3 CH3b>
1.500 C2H5>
H H 2(CH2ub>)2
CH-NHCH3
CH3 CH3b>
1.501 C2H5>
H H 0(CH2ub>)2
CH-NHC2H5
CH3 CH3
1.502 C2H5
H H 2(CH2)2
CH-NHC2H5
CH3 CH3
1.503 C2H5
H H 0(CH2)2
CH-N(CH3)2
CH3 CH3
1.504 C2H5
H H 2(CH2)2
CH-N(CH3)2
CH3 CH3
1.505 C2H5
H H 0(CH2)2
CH-NHOC2H5
CH3 CH3
1.506 C2H5
H H 2(CH2)2
CH-NHOC2H5
CH3 CH3
1.507 C2H5
H H 0(CH2)2
CH-N(CH3)OC2H5
CH3>
CH3
1.508> C2H5 H H
2(CH2)2 CH-
N(CH3)OC2H5 CH3>
CH3
1.509> C2H5 H H
0(CH2)2 C＝N-
NH CH3 CH3
> 1.510 C2H5
H H 2(CH2)2>
C＝N-
NH2 CH3 CH3
> 序号
R15 R16 R<
sup>17 n X Y L
M
1.511> C2H5 H H
0(CH2)2C＝N-
N(CH3)2 CH3
CH3
1.512 C2H5
H H 2(CH2)2
C＝N-N(CH3)2
CH3 CH3
1.513 C2H5
H H 0(CH2)2
C(CH3)-OCH3
CH3 CH3>
1.514 C2H5 H H 2(CH2b>)2
C(CH3)-OCH3
CH3 CH3>
1.515 C2H5 H H 0(CH2b>)2
O CH3 CH3
1.516 C2H5
H H 2(CH2)2
O CH3entry> CH3
1.517 CH3
CH3 H 0(CH2)2CH-NHCH3
Cl Cl
y> 1.518 CH3 CH3
H 2(CH2)2<
entry>CH-
NHCH3 Cl Cl
|
y> 1.519 CH3 CH3
H 0(CH2)2<
entry>CH-
NHC2H5 Cl Cl
> 1.520 CH3 CH3ub>
H 2(CH2)2b>
CH-
NHC2H5 Cl Cl
> 1.521 CH3 CH3ub>
H 0(CH2)2b>
CH-
N(CH3)2 Cl Cl
> 1.522 CH3 CH3ub>
H 2(CH2)2b>
CH-
N(CH3)2 Cl Cl
> 1.523 CH3 CH3ub>
H 0(CH2)2b>
CH-
NHOC2H5 Cl Cl
w> 1.524 CH3 CH3<
/sub> H 2(CH2)2ub>
CH-
NHOC2H5 Cl Cl
w> 1.525 CH3 CH3<
/sub> H 0(CH2)2ub>
CH-
N(CH3)OC2H5 Cly> Cl
|
1.526 CH3ntry> CH3 H 2(CH
2)2CH-
N(CH3)OC2H5 Cly> Cl
1.527 CH3ntry> CH3 H 0(CH
2)2C＝N-
NH2 Cl Cl
1.528
CH3 CH3ry> H 2(CH2)2y>C＝N-
NH2 Cl Cl
1.529
CH3 CH3ry> H 0(CH2)2y>C＝N-
N(CH3)2 Cl Cl
> 1.530 CH3 CH3ub>
H 2(CH2)2b>
C＝N-
N(CH3)2 Cl Cl
> 1.531 CH3 CH3ub>
H 0(CH2)2b>
C(CH3)-
OCH3 Cl Cl
1.532
CH3 CH3try> H 2(CH2)2y>C(CH3)-
OCH3 Cl Cl
|
1.533
CH3 CH3try> H 0(CH2)2y>O Cl Cl
|
1.534 CH3 CH3 H
2(CH2)2O<
entry> Cl Cl
1.535 Cb>2H5
H H 0y>(CH2)2CH-
NHCH3
Cl Cl
y> 1.536 C2H5 Hntry> H 2(CH2)2try>CH-
NHCH3 Cl Cl
|
y> 1.537 C2H5 Hntry> H 0(CH2)2try>CH-
NHC2H5 Cl Cl
> 1.538 C2H5
H H 2(CH2)2>
CH-
NHC2H5 Cl Cl
> 1.539 C2H5
H H 0(CH2)2>
CH-
N(CH3)2 Cl Cl
> 1.540 C2H5
H H 2(CH2)2>
CH-
N(CH3)2 Cl Cl
> 1.541 C2H5
H H 0(CH2)2>
CH-
NHOC2H5 Cl Cl
w> 1.542 C2H5> H H 2(CH2)2b>
CH-
NHOC2H5 Cl Cl
w> 1.543 C2H5> H H 0(CH2)2b>
CH-
N(CH3)OC2H5 Cly> Cl
1.544 C2H5ub>
H H 2(CH2
)2CH-
N(CH3)OC2H5 Cly> Cl
1.545 C2H5ub>
H H 0(CH2
)2C＝N-
NH2 Cl Cl
|
1.546
C2H5 H> H 2(CH2)2
C＝N-
NH2 Cl Cl
1.547
C2H5 H> H 0(CH2)2
C＝N-
N(CH3)2 Cl Cl
>
spec>> 序号
R15 R16 R
17 n X Y
L M
|
1.548y> C2H5 H H> 2(CH2)2C＝N-
N(CH3)2 Cl Cl
> 1.549 C2H5
H H 0(CH2)2>
C(CH3)-
OCH3 Cl Cl
1.550
C2H5 Hy> H 2(CH2)2>C(CH3)-
OCH3 Cl Cl
|
1.551
C2H5 Hy> H 0(CH2)2>O Cl Cl
|
1.552 C2H5 H H<
entry> 2(CH2)2Ontry> Cl Cl
1.553 CHb>3
CH3 H 0y>(CH2)2C＝
O
Cl Cl
1.554ntry> CH3 CH3 Hntry> 2(CH2)2C＝
O Cl Cl
1.555ntry> CH3 CH3 Hntry> 0(CH2)2CHOCH
3 Cl Cl
1.556try> CH3 CH3 Htry> 2(CH2)2CHOC
H3
Cl Cl
1.557
CH3 CH3> H 0(CH2)2
CHOC2H5 Cl Cl
w> 1.558 CH3 CH3<
/sub> H 2(CH2)2ub>
CHOC2H5 Clntry> Cl
1.559 CH3 CH3 H 0(CH>2)2
CHOiPr Cl Cl
1.560 CH3 CH3
H 2(CH2b>)2
CHOiPr Cl Cl>
1.561 CH3 CHb>3
H 0(CH2)>2
CHOH Cl Cl
<row> 1.562 CH3 CH3>
H 2(CH2)2
CHOH Cl Cltry> 1.563 CH3 CH3> H 0(CH2)2
C＝
NOCH3
Cl Cl
|
y> 1.564 CH3CH3<
entry> H 2(CH2)2ntry>C＝
NOCH3 Cl Cl
|
y> 1.565 CH3 CH3
H 0(CH2)2<
entry>C＝
NOC2H5 Cl Cl
> 1.566 CH3 CH3ub>
H 2(CH2)2b>
C＝
NOC2H5 Cl Cl
> 1.567 CH3 CH3ub>
H 0(CH2)2b>
C＝
NOiPr Cl Cl
|
1.568y> CH3 CH3 Hy> 2(CH2)2C＝
NOiPr
Cl Cl
1.569y> CH3 CH3 Hy> 0(CH2)2C＝
NOCH2CH＝
CHCl
Cl Cl
1.570> CH3 CH3 H> 2(CH2)2C＝
NOCH2CH＝
CHCl
Cl Cl
1.571> CH3 CH3 H> 0(CH2)2C＝
NOCH2C6H5
Cl> Cl
1.572 CH3try> CH3 H 2(CH2
)2C＝
NOCH2C6H5 Cl> Cl
1.573 CH3try> CH3 H 0(CH2
)2C(CH3)2y> Cl Cl
1.574 CH
3 CH3 H 2
(CH2)2C(CH3)2sub>
Cl Cl 1.575> C2H5 H H
0(CH2)2C＝
O
Cl Cl
1.576ntry> C2H5 H Hry> 2(CH2)2C＝
O Cl Cl
1.577ntry> C2H5 H Hry> 0(CH2)2CHOCH3
Cl Cl
1.578y> C2H5 H H> 2(CH2)2CHOCHub>3
Cl Cl
1.579
C2H5 H Hentry> 0(CH2)2CHO
C2H5
Cl Cl<
row> 1.580 C2H5 H
H 2(CH2)2<
/entry>CHOC2H5 Cl
Cl 1.581 C2H5
H H 0(CH2b>)2
CHOiPr ClCl> 1.582 C2H5
H H 2(CH2)>2
CHOiPr Cl Cl
1.583 C2H5
H
H 0(CH2)2>
CHOH Cl Clntry> 1.584 C2H5 H
H 2(CH2)2<
entry>CHOH Cl Cl
|
</table>ec> 序号 R15 R16 R<sup>17
n X Y L M
1.585> C2H5 H H
0(CH2)2C＝
NOCH3 Cl Cl
y> 1.586 C2H5 Hntry> H 2(CH2)2try>C＝
NOCH3 Cl Cl
|
y> 1.587 C2H5 Hntry> H 0(CH2)2try>C＝
NOC2H5 Cl Cl
> 1.588 C2H5
H H 2(CH2)2>
C＝
NOC2H5 Cl Cl
> 1.589 C2H5
H H 0(CH2)2>
C＝
NOiPr Cl Cl
|
1.590y> C2H5 H H> 2(CH2)2C＝
NOiPr
Cl Cl
1.591y> C2H5 H H> 0(CH2)2C＝
NOCH2CH＝
CHCl
Cl Cl
1.592> C2H5 H H
2(CH2)2C＝
NOCH2CH＝
CHCl
Cl Cl
1.593> C2H5 H H
0(CH2)2C＝
NOCH2C6H5
Cl> Cl
1.594 C2H5b>
H H 2(CH2sub>)2
C＝NOCH2C6H5
Cl> Cl
1.595 C2H5b>
H H 0(CH2sub>)2
C(CH3)2 Cl
Cl
1.596 C2ub>H5
H H 2ry>(CH2)2C(CH3)2>
Cl Cl
1.597ntry> CH3 CH3 Hntry> 0(CH2)2C＝
O CH3 CH3
<row> 1.598 CH3 CH3>
H 2(CH2)2
C＝
O CH3 CH3<
row> 1.599 CH3 CH3>
H 0(CH2)2
CHOCH3 CH3y> CH3 1.600 CH3sub>
CH3 H 2ntry>(CH2)2CHOCH3<
entry> CH3 CH3
> 1.601 CH3 CH3ntry> H 0(CH2)2try>CHOC2H5 CH3try> CH3
|
1.602 CH3
CH3 H 2<
entry>(CH2)2CHOC2H5<
/sub> CH3 CH3
w> 1.603 CH3 CH3<
/sub> H 0(CH2)2ub>
CHOiPr CH3 CH>3
1.604 CH3> CH3 H 2(CHub>2)2
CHOiPr CH3entry> CH3
1.605 C
H3 CH3 H 0
(CH2)2CHOH> CH3 CH3 1.
606 CH3 CH3> H 2(CH2)2
CHOH CH3 CH3
ow> 1.607 CH3 CH3
H 0(CH2)2<
/sub>C＝
NOCH3 CH3 CH3b>
1.608 CH3y> CH3 H 2(CH2sub>)2
C＝
NOCH3 CH3 CH3b>
1.609 CH3y> CH3 H 0(CH2sub>)2
C＝
NOC2H5 CH3
CH3
1.610 CH3>
CH3 H 2>(CH2)2C＝
NOC2H5 CH3
CH3
1.611 CH3>
CH3 H 0>(CH2)2C＝
NOiPr CH3 CH3
w> 1.612 CH3 CH3<
/sub> H 2(CH2)2ub>
C＝
NOiPr CH3 CH3
w> 1.613 CH3 CH3<
/sub> H 0(CH2)2ub>
C＝NOCH2CH＝
CHCl CH3 CH3
w> 1.614 CH3 CH3<
/sub> H 2(CH2)2ub>
C＝NOCH2CH＝
CHCl CH3 CH3
w> 1.615 CH3 CH3<
/sub> H 0(CH2)2ub>
C＝
NOCH2C6H5 CH3
CH3
1.616
CH3 CH3 H
2(CH2)2C＝
NOCH2C6H5 CH3
CH3 1.617
CH3 CH3 H
0(CH2)2C(CH3
)2 CH3 CH3ntry> 1.618 CH3 C
H3
H 2(CH2
)2C(CH3)2 CH<
sub>3 CH3 1.619ntry> C2H5 H Hry> 0(CH2)2C＝
O
CH3 CH3
<
row> 1.620 C2H5 H
H 2(CH2)2<
/entry>C＝
O CH3 CH3<
row> 1.621 C2H5 H
H 0(CH2)2<
/entry>CHOCH3 CH3> CH3
c> 序号 R15 R16 R17
n X Y L
M
1.622y> C2H5 H H> 2(CH2)2CHOCH3sub>
CH3 CH3
> 1.623 C2H5
H H 0(CH2)2>
CHOC2H5 CH3>
CH3
1.624> C2H5 H H
2(CH2)2CHOC2>H5
CH3 CH3<
/entry>
1.625 C2H5ntry> H H 0(CH2)
2
CHOiPr CH3> CH3
1.626 C2>H5
H H 2>(CH2)2CHOiPr CH3
CH3
1.627<entry> C2H5 H Hntry> 0(CH2)2CHOH> CH3 CH3
try> 1.628 C2H5 H<
entry> H 2(CH2)2ntry>CHOH CH3 CH3y>
|
1.629 C2H5> H H 0(CH2)b>2
C＝
NOCH3
CH3 CH3b>
1.630 C2H5>
H H 2(CH2ub>)2
C＝NOCH3
CH3 CH3b>
1.631 C2H5>
H H 0(CH2ub>)2
C＝NOC2H5
CH3 CH3
1.632 C2H5
H H 2(CH2)2
C＝NOC2H5
CH3 CH3
1.633 C2H5
H H 0(CH2)2
C＝NOiPr
CH3 CH3w> 1.634 C2H5> H H 2(CH2)2b>
C＝
NOiPr CH3 CH3
w> 1.635 C2H5> H H 0(CH2)2b>
C＝NOCH2CH＝
CHCl CH3 CH3
w> 1.636 C2H5> H H 2(CH2)2b>
C＝NOCH2CH＝
CHCl CH3 CH3
w> 1.637 C2H5> H H 0(CH2)2b>
C＝
NOCH2C6H5 CH3
CH3
1.638
C2H5 H H 2
(CH2)2C＝
NOCH2C6H5 CH3
CH3
1.639
C2H5 H H 0
(CH2)2C(CH3)
2 CH3 CH3try>
1.640 C2H5y> H H 2(CH2)ub>2
C(CH3)2 CHb>3
CH3
表2：下式化合物
<colspec> 序号R15 R16 R<sup>17
n X Y L M
2.1 CH3
CH3 H 0
N COCH3 Hntry> CH3
2.2 CH3 CH3 H 2<entry> N COCH3 H CHub>3
2.3 CH3y> CH3 H 0 Nntry> COC2H5 H CH
3
2.4 CH3ntry> CH3 H 2 N<
/entry> COC2H5 H C
H3
2.5 CH3</entry> CH3 H 0
N
COiPr H CH3</row> 2.6 CH3 CH3
H 2 N COiPrentry> H CH3
2.7</entry> C2H5 H Hntry> 0 N COCH3
H
CH3
2.8> C2H5 H H
2 N COCH3 Hntry> CH3
2.9 C2ub>H5
H H 0ry> N COC2H5 Hntry> CH3
2.10 C2</sub>H5
H H 2ntry> N COC2H5 H
CH3
2.11 C2
H5 H H 0 N COiPr H CH3<
/entry>
2.12 C2H5ntry> H H 2 N
COiPr
H CH3
> 2.13 CH3 CH3ntry> H 0 CH COCH3
ntry> H CH3
|
2.14 CH3 CH3 H 2 CH COCH3ntry> H CH3
2.15 CH3 CH3 H
0 CH COC2H5y> H CH3
2.16ntry> CH3 CH3 Hntry> 2 CH COC2H5
H CH3
2.17
CH3 CH3 H
0 CH COiPr Hry> CH3
2.18 CH<sub>3
CH3 H 2ntry> CH COiPr H CH3<
/sub>
2.19 C2H5ub>
H H 0 CH COCH3 H CH3ry>
2.20 C2H5> H H 2 CH C
OCH3
H CH3> 2.21 C2H5
H H 0 CH COC2
H5 H CH3
ow> 2.22 C2H5y> H H 2 CH COCb>2H5
H CH3>
2.23 C2H5
H H 0 CH CO
iPr H CH3
2.24
C2H5 H> H 2 CH COiPr Hntry> CH3
2.25 CH3
CH3 H 0 N COCH3 Hry> Cl
2.26 CH3<entry> CH3 H 2 N> COCH3 H Cl
w> 2.27 CH3 CH3<
/entry> H 0 N COC2b>H5
H Cl
2.28 CH3 CH3ry> H 2 N COC2H5
H Cl 2.29y> CH3 CH3 Hy> 0 N COiPr H> Cl
ec>ead> 序号
R15 R16 R
17 n X Y
L M
2.30> CH3 CH3 H> 2 NCOiPr H Cly>
2.31 C2H5 H H 0 NCOC
H3 H Cl
2.32
C2H5 H H
2 NCOCH3try> H Cl
2.33 C2H5 H H 0<entry> NCOC2H5 H
Cl
2.34 C2H5
H H 2 Ny>COC2H5 H Cltry>
2.35 C2H5> H H 0 NCOi
Pr
H Cl
2.36try> C2H5 H Hy> 2 NCOiPr H Cl
try>
2.37 CH3 CH<sub>3
H 0 CHCOCH3
H Cl
2.38
CH3 CH3y> H 2 CHCOCH3> H Cl
2.39 CH<sub>3
CH3 H 0ntry> CHCOC2H5 H
Cl
2.40 CH3>
CH3 H 2> CHCOC2H5 Htry> Cl
2.41 CH3ntry> CH3 H 0 CH>COiPr H Cl
2.42
CH3 CH3 H
2 CHCOiPr Hy> Cl
2.43 C2Hb>5
H H 0 CH</entry>COCH3 H Cl
> 2.44 C2H5
H
H 2 CHCOCH3
H Cl
2.45y> C2H5 H H> 0 CHCOC2H5ry> H Cl
2.46 C2H5
H H 2entry> CHCOC2H5
H
Cl
2.47 C2>H5
H H 0> CHCOiPr H Cl
2.48 C2H5 H> H 2 CHCOiPr> H
Cl
|
表3：下式
化合物
<colspec> 序号R15 R16 R<sup>17
n Y L M
3.1 CH3>
CH3 H 0> COCH3 H CH3
ow> 3.2 CH3 CH3<
/sub> H 2 COCH3
> H CH3
3.3y> CH3 CH3 Hy> 0 COC2H5 Hry> CH3
3.4 CHub>3
CH3 H 2try> COC2H5 H CH<
sub>3
3.5 CH3ry> CH3 H 0 COi
Pr
H CH3
3.6
CH3 CH3> H 2 COiPr H CHb>3
3.7 C2H5
H H 0 COCH3
H CH3
w> 3.8 C2H5 Hntry> H 2 COCH3
H
CH3 3.9> C2H5 H H
0 COC2H5 H> CH3
3.10 C2>H5
H H 2> COC2H5 H CH3b>
3.11 C2H5>
H H 0 COiPr> H CH3
3.12ry> C2H5 H H> 2 COiPr H CH3
3.13 CH3
CH3 H 0 COCH3sub>
H Cl 3.14
CH3 CH3 H
2 COCH3 H Clentry> 3.15 CH3 C
H3
H 0 COC2>H5
H Cl
3.16 CH3 CH3y> H 2 COC2H5ry> H Cl 3.17 CH>3
CH3 H 0> COiPr H Cl
3
.18 CH3 CH3> H 2 COiPr H Cl
ry> 3.19 C2H5> H H 0 COCH3<
/entry> H Cl
3.20y> C2H5 H H> 2 COCH3 H Cl
3.21 C2H5ntry> H H 0 COC2H>5
H Cl
3.22ntry> C2H5 H Hry> 2 COC2H5 Hntry> Cl
3.23 C2H
5 H H 0 C
OiPr H Cl 3.24
C2H5 H H<
entry> 2 COiPr H Cl
body>
表4：下式化合物
<colspec> 序号 R15 R16 R<sup>17
n X Y M
L
4.1> CH3 CH3 H> 0 CH2C＝
O H CH3
4.2
CH3 CH3 H
2 CH2C＝O
H CH3
4.3
CH3 CH3 H
0 CH2CHOCH3</sub>
H CH3
> 4.4 CH3 CH3ry> H 2 CH2CHOCH>3
H CH3
|
ntry> 4.5 CH3 CH3
H 0 CH2CHOC<
sub>2H5 H CH3y>
|
4.6 CH3 CH>3
H 2 CH2>CHOC2H5 H CHub>3
4.7 CH3> CH3 H 0 CHb>2
CHOiPr H CH3
4.8 CH3 CH3
H 2 CH2CHOiPr H CH3row> 4.9 CH3 CH3sub>
H 0 CH2ntry>CHOH H CH3
|
4.10 CH3 CH3ry> H 2 CH2CHO
H
H CH3
4.11
CH3 CH3 H
0 CH2C＝NOCH3
H CH3w> 4.12 CH3 CH3sub>
H 2 CH2ntry>C＝
NOCH3 H CH3
w> 4.13 CH3 CH3sub>
H 0 CH2ntry>C＝
NOC2H5 H CH3>
4.14 CH3
CH3 H 2 CH2>
C＝
NOC2H5 H CH3>
4.15 CH3
CH3 H 0 CH2>
C＝
NOiPr H CH3
y> 4.16 CH3 CH3ntry> H 2 CH2C＝
NOiPr H CH3
|
y> 4.17 CH3 CH3ntry> H 0 CH2C＝
NOCH2CH＝
CHCl H CH3
|
> 4.18 CH3 CH3try> H2 CH2C＝
NOCH2CH＝
CHCl H CH3
|
> 4.19 CH3 CH3try> H 0 CH2C＝
NOCH2C6H5 H
CH3
|
4.20 CH3>
CH3 H 2> CH2C＝
NOCH2C6H5 H
CH3
4.21 CH3>
CH3 H 0> CH2C(CH3)2
H CH3
4.22 CH3
CH3 H 2
CH2C(CH3)2 H CH3
4.23
C2H5 H H 0 CH2C＝O
H CH3
4.24
C2H5 H H
2 CH2C＝O
H CH3
4.25
C2H5 H H
0 CH2CHOCH3</sub>
H CH3
> 4.26 C2H5 Hy> H 2 CH2CHOCH>3
H CH3
|
ntry> 4.27 C2H5 H<
entry> H 0 CH2CHOCb>2H5
H CH3>
|
4.28 C2H5<entry> H H 2 CH2>CHOC2H5 H CHub>3
4.29 C2H>5
H H 0 CHub>2
CHOiPr H CH3>
>d> 序号
R15 R16R<
sup>17 n X Y
M L
4.30> C2H5 H H
2 CH2CHOiPr H
CH3
4.31 C2H5 H H 0<entry> CH2CHOH H CH
3
4.32 C2Hb>5
H H 2 CH<sub>2
CHOH H CH3>
4.33 C2H5entry> H H 0 CH2
C＝NOCH3
H CH3w> 4.34 C2H5
H H 2 CH2y>C＝
NOCH3 H CH3
w> 4.35 C2H5
H H 0 CH2y>C＝
NOC2H5 H CH3>
4.36 C2H5entry> H H 2 CH2
C＝NOC2H5
H CH3>
4.37 C2H5entry> H H 0 CH2
C＝NOiPr
H CH3
y> 4.38 C2H5 Htry> H 2 CH2C＝
NOiPr H CH3
|
y> 4.39 C2H5 Htry> H 0 CH2C＝
NOCH2CH＝
CHCl H CH3
|
> 4.40 C2H5 Hy> H 2 CH2C＝
NOCH2CH＝
CHCl H CH3
|
> 4.41 C2H5 Hy> H 0 CH2C＝
NOCH2C6H5 H
CH3
|
4.42 C2H5
H H 2 CH2
C＝NOCH2C6H5
H CH3
4.43 C2H5
H H 0 CH2
C(CH3)2 H
CH3
4.44 C2H5
H H 2 CH2C(CH3)2entry> H CH3
4.45</entry> CH3 CH3 H<
/entry> 0 CH2C＝
O
H Cl
4.46ry> CH3 CH3 Hry> 2 CH2C＝
O H Cl
4.47ry> CH3 CH3 Hry> 0 CH2CHOCH3
H Cl
4.48 CHub>3
CH3 H 2try> CH2CHOCH3 H
Cl
4.49 CH3>
CH3 H 0> CH2CHOC2H5> H Cl
4.50 CH3</sub>
CH3 H 2ntry> CH2CHOC2H5ntry> H Cl
4.51 CH>3
CH3 H 0> CH2CHOiPr H
Cl
4.52 CH3> CH3 H 2 CH2ub>
CHOiPr H Cl
> 4.53 CH3 CH3try> H 0 CH2CH
OH
H Cl 4.54ntry> CH3 CH3 Hntry> 2 CH2CHOH Htry> Cl
4.55 CH3ntry> CH3 H 0 C
H2
C＝
NOCH3 H Cl> 4.56 CH3 CH3try> H 2 CH2C＝
NOCH3 H Cl
|
> 4.57 CH3 CH3try> H 0 CH2C＝
NOC2H5 H Cl
|
> 4.58 CH3 CH3b>
H 2 CH2y>C＝
NOC2H5 H Cl
> 4.59 CH3 CH3b>
H 0 CH2y>C＝
NOiPr H Cl
4.60> CH3 CH3 H> 2 CH2C＝
NOiPr
H Cl
4.61> CH3 CH3 H> 0 CH2C＝
NOCH2CH＝
CHCl
H Cl
4.62
CH3 CH3 H
2 CH2C＝
NOCH2CH＝
CHCl H Cl
4.63
CH3 CH3 H
0 CH2C＝
NOCH2C6H5 H
Cl 4.64 CH3> CH3 H 2 CH2ub>
C＝
NOCH2C6H5 H
Cl
4.65 CH3> CH3 H 0 CH2ub>
C(CH3)2 Hy> Cl
4.66 CH3try> CH3 H 2 CH2<
/sub>C(CH3)2 Htry> Cl
lspec>
序号 R15 R16 R17
n X Y M
L
4.67y> C2H5 H H> 0 CH2C＝
O H Cl
4.68ntry> C2H5 H Hry> 2 CH2C＝
O H Cl
4.69ntry> C2H5 H Hry> 0 CH2CHOCH3
H Cl
4.70 Cub>2H5
H H 2try> CH2CHOCH3 H
Cl
4.71 C2>H5
H H 0> CH2CHOC2H5> H Cl
4.72 C2sub>H5
H H 2ntry> CH2CHOC2H5ntry> H Cl
4.73 C>2H5
H H 0> CH2CHOiPr H
Cl
4.74 C2H5 H H 2 CH2b>
CHOiPr H Cl
4.75 C2H5 Hy> H 0 CH2CHO
H
H Cl
|
4.76ntry> C2H5 H Hry> 2 CH2CHOH Hy> Cl
4.77 C2Hub>5
H H 0 CH2
C＝NOCH3
H Cl
> 4.78 C2H5 Htry> H 2 CH2C＝
NOCH3 H Cl
|
> 4.79 C2H5 Htry> H 0 CH2C＝
NOC2H5 H Cl
> 4.80 C2H5
H H 2 CH2>C＝
NOC2H5 H Cl
> 4.81 C2H5
H H 0 CH2>C＝
NOiPr H Cl
|
4.82> C2H5 H H
2 CH2C＝
NOiPr
H Cl
4.83> C2H5 H H
0 CH2C＝
NOCH2CH＝
CHCl
H Cl
4.84> C2H5 H H
2 CH2C＝
NOCH2CH＝
CHCl
H Cl
4.85> C2H5 H H
0 CH2C＝
NOCH2C6H5
H Cl
4.86 C2H5>
H H 2 CH2ub>
C＝NOCH2C6H5
H Cl
4.87 C2H5>
H H 0 CH2ub>
C(CH3)2 Hy> Cl
4.88 C2H5ub>
H H 2 CH2C(CH3)2 Hntry> Cl
4.89 CH3 CH3 H 0(CH>2)2
C＝
O H Cl
4.90ntry> CH3 CH3 Hntry> 2(CH2)2C＝
O H Cl
4.91ntry> CH3 CH3 Hntry> 0(CH2)2CHOCH
3 H Cl
4.92ry> CH3 CH3 Hry> 2(CH2)2CHOCH
3
H Cl
4.93
CH3 CH3 H
0(CH2)2CHOC2H5
H Cl> 4.94 CH3 CH3ub>
H 2(CH2)2b>
CHOC2H5 Hry> Cl
4.95 CH3<
entry> CH3 H 0(CH
2)2CHOiPr H Clentry>
4.96 CH3 CH3
H 2(CH2)2
CHOiPr H Clrow> 4.97 CH3 CH
3 H 0(CH2)2
CHOH H Cl
w> 4.98 CH3 CH3<
/entry> H 2(CH2)2entry>CHOH H Cl> 4.99
|
CH3 CH3ntry> H 0(CH2)2try>C＝
NOCH3 H Cl> 4.100 CH3 CH3
H 2(CH2)2<
entry>C＝
NOCH3 H Cl
|
> 4.101 CH3 CH3
H 0(CH2)2<
entry>C＝
NOC2H5 H Cl
> 4.102 CH3 CH3sub>
H 2(CH2)2ub>
C＝
NOC2H5 H Cl
> 4.103 CH3 CH3sub>
H 0(CH2)2ub>
C＝
NOiPr H Cl
|
olspec> 序号R15 R16 R<sup>17
n X Y M
L
4.104y> CH3 CH3 Hy> 2(CH2)2C＝
NOiPr H Cl
4.105> CH3 CH3 H> 0(CH2)2C＝
NOCH2CH＝
CHCl
H Cl
4.106> CH3 CH3 H> 2(CH2)2C＝
NOCH2CH＝
CHCl
H Cl
4.107> CH3 CH3 H> 0(CH2)2C＝
NOCH2C6H5
H
Cl
4.108 CH3y> CH3 H 2(CH2sub>)2
C＝
NOCH2C6H5 H
Cl
4.109 CH3y> CH3 H 0(CH2sub>)2
C(CH3)2
H Cl
4.110 CH3sub>
CH3 H 2ntry>(CH2)2C(CH3)2b>
H Cl
4.111<entry> C2H5 H Hntry> 0(CH2)2C＝
O H Cl
4.112ntry> C2H5 H Hry> 2(CH2)2C＝
O H Cl
4.113ntry> C2H5 H Hry> 0(CH2)2CHOCH3
H Cl
4.114y> C2H5 H H> 2(CH2)2CHOCHub>3
H Cl
4.115</entry> C2H5 H Hntry> 0(CH2)2CHOC
2H5
H Cl
w> 4.116 C2H5 Hentry> H 2(CH2)2ntry>CHOC2H5 H Cl
4.117 C2H5entry> H H 0(CH2
)2
CHOiPr H Clrow> 4.118 C2H5ry> H
H 2(CH2)2sub>
CHOiPr H Cl> 4.119 C2H5 Htry> H 0(CH2)2y>CHOH H Cl 4
.120
C2H5 H
H
2(CH2)2C
HOH H Cl 4.121> C2H5 H H
0(CH2)2C＝
NOCH3
H Cl
> 4.122 C2H5 Htry> H 2(CH2)2y>C＝
NOCH3 H Cl
|
> 4.123 C2H5 Htry> H 0(CH2)2y>C＝
NOC2H5 H Cl
|
> 4.124 C2H5
H H 2(CH2)2>
C＝
NOC2H5 H Cl
> 4.125 C2H5
H H 0(CH2)2>
C＝
NOiPr H Cl 4.126> C2H5 H H
2(CH2)2C＝
NOiPr
H Cl
4.127> C2H5 H H
0(CH2)2C＝
NOCH2CH＝
CHCl
H Cl
4.128> C2H5 H H
2(CH2)2C＝
NOCH2CH＝
CHCl
H Cl
4.129> C2H5 H H
0(CH2)2C＝
NOCH2C6H5
H
Cl 4.130 C2H5>
H H 2(CH2ub>)2
C＝
NOCH2C6H5 H
Cl 4.131 C2H5>
H H 0(CH2ub>)2
C(CH3)2
H Cl 4.132 C2b>H5
H H 2y>(CH2)2C(CH3)2
H Cl
4.133ry> CH3 CH3 Hry> 0(CH2)2C＝
O H CH3
4.
134 CH3 CH3> H 2(CH2)2
C＝
O H CH3 4.
135 CH3 CH3> H 0(CH2)2
CHOCH3 H CH3
ow> 4.136 CH3 CH3
H 2(CH2)2<
/sub>CHOCH3 H CHb>3
4.137 CH3y> CH3 H 0(CH<
sub>2)2
CHOC2H5y> H CH3
4.138ntry> CH3 CH3 Hntry> 2(CH2)2CHOC
2H5
H CH3try>
4.139 CH3 CH
3 H 0(CH2)<
sub>2CHOiPr H CH3b>
4.140 CH3y> CH3 H 2(CH2sub>)2
CHOiPr H CH>3
<colspec>c> 序号R15 R16Rup>17
n X Y M L
4.141> CH3 CH3 H> 0(CH2)2CHOHntry> H CH3
4.142 CH3 CH3 H
2(CH2)2CHOHry> H CH3
4.143ntry> CH3 CH3 Hntry> 0(CH2)2C＝
NOCH3
H CH3
w> 4.144 CH3 CH3<
/sub>
H 2(CH2)2ub>
C＝NOCH3
H CH3w> 4.145 CH3 CH3<
/sub> H 0(CH2)2ub>
C＝
NOC2H5 H CH3>
4.146 CH3> CH3 H 2(CH2ub>)2
C＝
NOC2H5 H CH3>
4.147 CH3> CH3 H 0(CH2ub>)2
C＝
NOiPr H CH3
y> 4.148 CH3 CH3
H 2(CH2)2<
entry>C＝
NOiPr H CH3
|
y> 4.149 CH3 CH3
H 0(CH2)2<
entry>C＝NOCH2CH＝
CHCl H CH3
|
> 4.150 CH3 CH3ntry> H 2(CH2)2try>C＝NOCH2CH＝
CHCl H CH3
|
> 4.151 CH3 CH3ntry> H 0(CH2)2try>C＝
NOCH2C6H5 H
CH3
|
4.152 CH3b>
CH3 H 2y>(CH2)2C＝
NOCH2C6H5 H
CH3
4.153 CH3b>
CH3 H 0y>(CH2)2C(CH3)2
H CH3
4.154
CH3 CH3 H
2(CH2)2C(CH3)2
H CH3</entry>
4.155 C2H5ntry> H H 0(CH2)
2
C＝O
H CH3
4.156
C2H5 H H
2(CH2)2C＝
O
H CH3
4.157
C2H5 H H
0(CH2)2CHOCH3
H CH3w> 4.158 C2H5> H H 2(CH2)2b>
CHOCH3 H CH3
4.159 C2H5sub>
H H 0(CH2
)2CHOC2H5ry> H CH3
4.160ntry> C2H5 H Hry> 2(CH2)2CHOC2sub>H5
H CH3
w> 4.161 C2H5> H H 0(CH2)2b>
CHOiPr H CH3
>
4.162 C2H5
H H 2(CH2)>2
CHOiPr H CH3
4.163 C2H5entry> H H 0(CH2
)2
CHOH H CH3ub>
4.164 C2H5>
H H 2(CH2ub>)2
CHOH H CH3
4.165 C2H5 H H 0(CH>2)2
C＝NOCH3
H CH3w> 4.166 C2H5> H H 2(CH2)2b>
C＝
NOCH3 H CH3
w> 4.167 C2H5> H H 0(CH2)2b>
C＝
NOC2H5 H CH3>
4.168 C2H5
H H 2(CH2b>)2
C＝
NOC2H5 H CH3>
4.169 C2H5
H H 0(CH2b>)2
C＝
NOiPr H CH3
y> 4.170 C2H5 Hntry> H 2(CH2)2try>C＝
NOiPr H CH3
|
y> 4.171 C2H5 Hntry> H 0(CH2)2try>C＝NOCH2CH＝
CHCl H CH3
|
> 4.172 C2H5 Htry> H 2(CH2)2y>C＝NOCH2CH＝
CHCl H CH3
|
> 4.173 C2H5 Htry> H 0(CH2)2y>C＝
NOCH2C6H5 H
CH3
|
4.174 C2H5
H H 2(CH2)2
C＝NOCH2C6H5
H CH3
4.175 C2H5
H H 0(CH2)2
C(CH3)2ntry> H CH3
4.176 C2H5 H Hentry> 2(CH2)2C(CH
3)2
H CH3ry>
4.177 CH3 CH<sub>3
p-CH3-C6H4-SO2-
0(CH2)2C＝
O
H CH3
>
lspec> 序号R15 R16 R<sup>17
nX Y M L
4.178> CH3 CH3 p-
CH3-C6H4-SO2-
2(CH2)2C＝
O H CH3
4.179
CH3 CH3> p-CH3-C6H4-SO2-
0(CH2)2CH
OCH3 H CH3
> 4.180 CH3 CH3ub>
p-CH3-C6H4-
SO2-
2(CH2)2CH
OCH3 H CH3
> 4.181 CH3 CH3ub>
P-CH3-C6H4-
SO2-
0(CH2)2CH
OC2H5 H CH3
4.182 CH3 CH3
p-CH3-C6H4-SO2-
2(CH2)2CHOC2H5
H CH3
4.183 CH3 CH3
p-CH3-C6H4-SO2-
0(CH2)2CHOiPr
H CH3
4.184
CH3 CH3try> p-CH3-C6H4-SO2-
2(CH2)2CH
OiPr H CH3
|
4.185
CH3 CH3try> p-CH3-C6H4-SO2-
0(CH2)2CH
OH H CH3
|
4.186
CH3 CH3ry> p-CH3-C6H4-SO2-
2(CH2)2CH
OH H CH3
4.187
CH3 CH3ry> p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH3 H CH3
w> 4.188 CH3 CH3<
/sub> p-CH3-C6H4-
SO2-
2(CH2)2C＝
NOCH3 H CH3
w> 4.189 CH3 CH3<
/sub> p-CH3-C6H4-
SO2-
0(CH2)2C＝
NOC2H5 H CH3>
4.190 CH3> CH3 p-CH3-
C6H4-SO2-
2(CH2)2C＝
NOC2H5 H CH3>
4.191 CH3> CH3 p-CH3-
C6H4-SO2-
0(CH2)2C＝
NOiPr H CH3
y> 4.192 CH3 CH3
p-CH3-C6H4-SO2-
2(CH2)2C＝
NOiPr H CH3
|
y> 4.193 CH3 CH3
p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH2CH＝
CHCl H CH3
|
> 4.194 CH3 CH3ntry> P-CH3-C6H4-SC2-
2(CH2)2C＝
NOCH2CH＝
CHCl H CH3
|
> 4.195 CH3 CH3ntry> p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH2C6H5 H
CH3
|
4.196 CH3b>
CH3 p-CH3-C6H4-SO2-
2(CH2)2C＝NOCH2C6H5
H CH3
4.197 CH3b>
CH3 p-CH3-C6H4-SO2-
0(CH2)2C(CH3)2
H CH3ntry>
4.198 CH3 CH3
P-CH3-C6H4-SO2-
2(CH2)2C(CH3)2
H CH3ntry>
4.199 C2H5ry> H p-CH3-C6H4-
SO2-
0(CH2)2C＝O
H CH3
4.200
C2H5 H p-CH3-C6H4-SO2-
2(CH2)2C＝O
H CH3
4.201
C2H5 H P-CH3-C6H4-SO2-
0(CH2)2CHOCH3
H CH3> 4.202 C2H5
H P-CH3-C6H4-
SO2-
2(CH2)2CH
OCH3 H CH3
> 4.203 C2H5
H p-CH3-C6H4-
SO2-
0(CH2)2CH
OC2H5 H CH3
4.204 C2H5entry> H p-CH3-C6H4-
SO2-
2(CH2)2CHOC2H5
H CH3
4.205 C2H5entry> H p-CH3-C6H4-
SO2-
0(CH2)2CHOiPr
H CH3
4.206
C2H5 Hy> P-CH3-C6H4-SO2-
2(CH2)2CH
OiPr H CH3
|
4.207
C2H5 Hy> P-CH3-C6H4-SO2-
0(CH2)2CH
OH H CH3
|
4.208
C2H5 H> p-CH3-C6H4-SO2-
2(CH2)2CH
OH H CH3
4.209
C2H5 H> p-CH3-C6H4-SO2-
0(CH2)2C＝
NOCH3 H CH3
w> 4.210 C2H5> H p-CH3-C6H4-
SO2-
2(CH2)2C＝
NOCH3 H CH3
w> 4.211 C2H5> H p-CH3-C6H4-
SO2-
0(CH2)2C＝
NOC2H5 H CH3>
4.212 C2H5
H p-CH3-
C6H4-SO2-
2(CH2)2C＝
NOC2H5 H CH3>
4.213 C2H5
H P-CH3-
C6H4-SO2-
0(CH2)2C＝
NOiPr H CH3
y> 4.214 C2H5 Hntry> p-CH3-C6H4-SO2-
2(CH2)2C＝
NOiPr H CH3
|
group>
c> 序号R15R16 Rup>17
n X Y M L
4.215> C2H5 H p-
CH3-C6H4-SO2-
0(CH2)2 C
＝NOCH2CH＝
CHCl H CH3
> 4.216 C2H5 Htry> p-CH3-C6H4-SO2-
2(CH2)2 C
＝NOCH2CH＝
CHCl H CH3
|
> 4.217 C2H5 Htry> p-CH3-C6H4-SO2-
0(CH2)2 C
＝
NOCH2C6H5 H
CH3
|
4.218 C2H5
H p-CH3-C6H4-SO2-
2(CH2)2 C＝
NOCH2C6H5
H CH3
4.219 C2H5
H p-CH3-C6H4-SO2-
0(CH2)2 C(CH3)2
H CH3entry>
4.220 C2H5try> H p-CH3-C6H4-
SO2-
2(CH2)2 C(CH3)2
H CH3entry>
4.221 CH3 CH3
H0(CH2)2
CH-NHCH3
H CH3w> 4.222 CH3 CH3<
/sub> H2(CH2)2ub>
CH-
NHCH3 H CH3
w> 4.223 CH3 CH3<
/sub> H0(CH2)2ub>
CH-
NHC2H5 H CH3>
4.224 CH3> CH3 H2(CH2b>)2
CH-
NHC2H5 H CH3>
4.225 CH3> CH3 H0(CH2b>)2
CH-
N(CH3)2 H CH3>
4.226 CH3> CH3 H2(CH2b>)2
CH-
N(CH3)2 H CH3>
4.227 CH3> CH3 H0(CH2b>)2
CH-
NHOC2H5 H CH3b>
4.228 CH3y> CH3 H2(CH2ub>)2
CH-
NHOC2H5 H CH3b>
4.229 CH3y> CH3 H0(CH2ub>)2
CH-
N(CH3)OC2H5 Hy> CH3
4.230 CH3sub>
CH3 H2try>(CH2)2 CH-
N(CH3)OC2H5 Hy> CH3
4.231 CH3sub>
CH3 H0try>(CH2)2 C＝N-
NH2 H CH3
<row> 4.232 CH3 CH3>
H2(CH2)2
C＝N-
NH2 H CH3<
row> 4.233 CH3 CH3>
H0(CH2)2
C＝N-
N(CH3)2 H CH3>
4.234 CH3> CH3 H2(CH2b>)2
C＝N-
N(CH3)2 H CH3>
4.235 CH3> CH3 H0(CH2b>)2
C(CH3)-
OCH3 H CH3
> 4.236 CH3 CH3ub>
H2(CH2)2b>
C(CH3)-
OCH3 H CH3
> 4.237 CH3 CH3ub>
H0(CH2)2b>
O H CH3w> 4.238 CH3 CH3<
/sub> H2(CH2)2ub>
O H CH3
ow> 4.239 C2H5y> H H0(CH2)2ub>
CH-
NHCH3 H CH3
w> 4.240 C2H5> H H2(CH2)2b>
CH-
NHCH3 H CH3
w> 4.241 C2H5> H H0(CH2)2b>
CH-
NHC2H5 H CH3>
4.242 C2H5
H H2(CH2>)2
CH-
NHC2H5 H CH3>
4.243 C2H5
H H0(CH2>)2
CH-
N(CH3)2 H CH3>
4.244 C2H5<
/entry> H H2(CH2
)2 CH-
N(CH3)2 H CH3>
4.245 C2H5
H H0(CH2>)2
CH-
NHOC2H5 H CH3b>
4.246 C2H5>
H H2(CH2ub>)2
CH-
NHOC2H5 H CH3b>
4.247 C2H5>
H H0(CH2ub>)2
CH-
N(CH3)OC2H5 Hy> CH3 4.248 C2b>H5
H H2y>(CH2)2 CH-
N(CH3)OC2H5 Hy> CH3
4.249 C2b>H5
H H0y>(CH2)2 C＝N-
NH2 H CH3
<
row> 4.250 C2H5 H
H2(CH2)2entry> C＝N-
NH2
H CH3<
row> 4.251 C2H5 H
H0(CH2)2entry> C＝N-
N(CH3)2
H CH3>
>d> 序号
R15 R16 R<
sup>17 n X Y
M L
4.252y> C2H5 H H> 2(CH2)2 C＝N-
N(CH3)2 H CH3>
4.253 C2H5 H H 0(CH2b>)2
C(CH3)-OCH3
H CH3> 4.254 C2H5
H H 2(CH2)2>
C(CH3)-
OCH3 H CH3
> 4.255 C2H5
H H 0(CH2)2>
O H CH3
> 4.256 C2H5
H H 2(CH2)2>
O H CH3
> 4.257 CH3 CH3ub>
H 0(CH2)2b>
CH-
NHCH3 H Cl
> 4.258 CH3 CH3ntry> H 2(CH2)2try> CH-
NHCH3 H Cl
|
> 4.259 CH3 CH3ntry> H 0(CH2)5try> CH-
NHC2H5 H Cl
> 4.260 CH3 CH3ub>
H 2(CH2)2b>
CH-
|